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1-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)but-3-enamide
N-[3-(1H-imidazol-1-yl)propyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-(2,6-dimethylphenyl)-2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-amino-2-(morpholin-4-yl)-5-(4-oxo-4H-chromen-3-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-1-[(2S)-oxolan-2-ylmethyl]-4-phenyl-1H-imidazole
2-[2-(3-ethoxyphenyl)phenyl]ethan-1-amine
3-methyl-5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-pyrazole
3-[(4-methoxyphenyl)methyl]-1,8-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
[2-(6-methoxypyridin-2-yl)phenyl]methanol
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
methyl 2-[methyl({3-[(2,4,6-trimethylpyridin-3-yl)carbamoyl]phenyl}methyl)amino]acetate
N-({1-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
2-[(3-methoxyphenyl)amino]-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]butanamide
2-fluoro-N-methyl-5-({[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]carbamoyl}amino)benzamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]propanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propan-1-one
{1-[(E)-2-phenylethenesulfonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
(cyclohexylmethyl)({[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl})amine
3-(1H-pyrazol-1-ylmethyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
2-methoxy-N-[4-methyl-3-({[3-methyl-1-(pyridin-3-yl)butyl]carbamoyl}amino)phenyl]acetamide
2-[2-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)phenoxy]acetic acid
N-{1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[2-(1H-imidazol-1-yl)ethyl]-3-[(pyridin-2-ylmethyl)sulfamoyl]benzamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-[(diethylamino)methyl]-5-ethylfuran-2-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-N-[(3-methyloxetan-3-yl)methyl]-1,3-oxazole-4-carboxamide
3-(1,3-benzothiazol-6-yl)-1-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]urea
4-chloro-1-methyl-3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-1H-indazole
(3R,5S)-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-methyl-5-{[5-oxo-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}furan-2-carboxamide
3-methyl-3-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]urea
3-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
6-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2-methyl-4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(thiophen-2-yl)propan-1-one
1-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)azepan-2-one
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methoxypyridine
2-(5-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}furan-2-yl)benzonitrile
8-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(1H-imidazol-2-yl)benzamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)piperidin-2-one
(3R,4R)-4-(hydroxymethyl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
7-(2-oxopyrrolidin-1-yl)-4-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1,2,3,4-tetrahydroquinolin-2-one
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-(thiophen-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N,3,5-trimethyl-N-[2-(methylsulfanyl)ethyl]-1H-indole-2-carboxamide
2-tert-butyl-8-(2-methoxyquinoline-4-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene