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2-methyl-4-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]phenol
N-butyl-1-ethyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-cyclopropyl-1-[1-(3-methylbenzoyl)piperidin-4-yl]piperidine-4-carboxamide
5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2-dihydroquinolin-2-one
N-[1-(2-propoxyphenyl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
9-(2,3-difluoro-6-methoxybenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-3-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-N,N-dimethylfuran-2-carboxamide
1-butyl-4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-2-one
1-(prop-2-en-1-yl)-5-[(pyridin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidin-2-one
1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(3-methyl-1H-pyrazol-1-yl)acetamide
2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
1-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(propan-2-yl)urea
1-{4-[({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)amino]piperidin-1-yl}ethan-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-fluoro-2-methylbenzamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-methyl-1H-imidazol-1-yl)acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(oxane-2-carbonyl)piperidine-4-carboxamide
2-(morpholin-2-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]acetamide
ethyl 1-({3-[4-(methoxycarbonyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-2-carboxylate
5-cyclopropyl-N-ethyl-N-(2-hydroxyethyl)-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
ethyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
methyl (2S,4S)-1-(naphthalen-2-ylmethyl)-4-propanamidopyrrolidine-2-carboxylate
methyl({[1-(propan-2-yl)piperidin-3-yl]methyl}){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
5-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[1-(2-hydroxyethyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
6-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-(3-phenylpropyl)piperidine-3-carboxamide
N-[(3-fluorophenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(1H-indol-5-yl)-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}pyrrolidin-3-ol
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
3-methyl-7-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[3-(3-fluorophenyl)phenyl]-1-[(2-propylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
(3R,5S)-1-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3-carboxamide
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}piperidine
N-[4-(2,1,3-benzothiadiazol-4-yl)-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methylpropanamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
6-(benzyloxy)-1-(2-methylpropyl)-4-(thiophene-2-carbonyl)-1,4-diazepan-2-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[4-(4-methylpiperazin-1-yl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
3,5-dimethyl-4-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-1H-pyrrole-2-carboxylic acid
2-(ethylamino)-N-[1-(2-phenylethyl)piperidin-4-yl]pyrimidine-5-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)acetamide
3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]benzamide