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N-(1-methoxybutan-2-yl)-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
(5-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}furan-2-yl)methanol
2-[methyl(pyridin-4-ylmethyl)amino]-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-ethyl-N4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-methylpyrimidine-2,4-diamine
6-[(2-methylprop-2-en-1-yl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-(cyclobutylmethoxy)-5-[(1,2-oxazol-3-ylmethyl)carbamoyl]benzoic acid
4-{4-[2-(2-fluorophenyl)ethyl]-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}-1,4-diazepane-1-carbaldehyde
(2R,6R)-4-[3-(1H-pyrazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[4-(4-acetylphenyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
N'1-[(3R,4S)-1-(cyclohexylmethyl)-4-cyclopropylpyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
4-(4-ethenylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
3-(3-methoxyphenyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-5-carboxamide
2-[3-(2-methylphenoxy)azetidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3,5-difluoro-2-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridine
4-[({4-methyl-5-[1-(2-phenylpropyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5,6-dimethylpyridine-3-carboxamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[4-(pyridin-3-yloxy)phenyl]propanamide
N-(cyclopropylmethyl)-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
8-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1-benzothiophen-2-ylmethyl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclopentyl-3-{[(5-methylpyrazin-2-yl)methyl]sulfamoyl}benzamide
(4aS,8aR)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1H-indole-6-carboxamide
4-[4-(3-methoxypropyl)piperazine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N-benzyl-N-methyl-3-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
5-oxo-1-(2-propoxyethyl)pyrrolidine-3-carboxylic acid
5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-(3-phenylpropyl)piperidine-3-carboxylic acid
ethyl (4aS,8aR)-6-{imidazo[1,2-b]pyridazine-3-carbonyl}-decahydro-1,6-naphthyridine-4a-carboxylate
N-{[1-(2-chlorophenyl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}methanesulfonamide
N-(2-methoxy-5-phenylphenyl)-3-(piperidin-1-yl)azetidine-1-carboxamide
3-[(3R,4S)-1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-(pyrimidin-4-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
8-[1-(1H-imidazol-1-yl)propan-2-yl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(3-chlorophenyl)ethyl]-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidin-2-one
N-[(1-benzylpiperidin-4-yl)methyl]-1-(difluoromethyl)-N-methyl-1H-pyrazole-3-carboxamide
1-[1-(piperidine-1-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}-2-(furan-2-yl)pyrimidine
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidin-3-yl]cyclopropanecarboxamide
7-(6-chloro-2-methylquinoline-4-carbonyl)-2-methyl-2,7-diazaspiro[4.5]decane
2-(morpholin-4-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
N-methyl-2-({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)acetamide
(1R,5R)-6-benzyl-3-(6-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3-methylphenyl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
3-(4-hydroxyphenyl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]propan-1-one
5-[3-(2-methylphenyl)piperidine-1-carbonyl]pyridin-2-amine
2-(4-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-6-phenyl-3,4-dihydropyrimidin-4-one
5-methyl-4-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(prop-2-en-1-yl)-1H-pyrazole
4-[1-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1H-imidazol-2-yl]phenol