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3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5,6-dimethylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methoxyphenyl)methyl]acetamide
1-ethyl-N-[2-(3-fluorophenyl)ethyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(pyridin-2-ylsulfanyl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}ethan-1-one
methyl (1R,3S,3aR,6aS)-1-benzyl-3-(2-hydroxyphenyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(3S,4R)-1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
4-(1-butyl-1H-imidazol-2-yl)-1-(2,6-dimethoxybenzoyl)piperidine
4-(hydroxymethyl)-1-[5-(methoxymethyl)thiophene-2-carbonyl]azepan-4-ol
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-propanoylpiperidine-3-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-methoxypyrimidin-4-amine
1-(2,5-dimethylfuran-3-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-(4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetic acid
2-(adamantan-1-yl)-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]acetamide
1-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxylic acid
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-3-yl)acetamide
1-(5-tert-butyl-2-methoxyphenyl)-3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]urea
4-[4-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(3-hydroxy-3-methylbutyl)-N-(2-methylpropyl)-N-(pyridin-4-ylmethyl)benzamide
N-[1-(thian-4-yl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,4S)-5-(1-aminocyclopropanecarbonyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
[(2S,4R)-4-(dimethylamino)-1-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-2-yl]methanol
9-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
N-[(3S,4R)-1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
6-methyl-1-[2-(methylsulfanyl)phenyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-one
2-(cyclopropylmethyl)-9-[2-(4-hydroxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-1H-1,2,4-triazole-5-carboxamide
3-[(dimethylamino)methyl]-1-{[4-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-ol
3-methyl-4-({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)piperazin-2-one
4-[(4-methoxyphenyl)methyl]-1-(naphthalene-1-carbonyl)-1,4-diazepan-5-one
(3aR,6aR)-2-methanesulfonyl-5-[2-(4-methoxyphenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2,5-dimethylphenyl)-4-(oxan-4-yl)piperazine-1-carboxamide
2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carboxamide
4,6-dimethyl-3-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[2-(morpholin-4-yl)propyl]pyrimidine-5-carboxamide
[(2-fluoro-3-methoxyphenyl)methyl](methyl)(thiophen-3-ylmethyl)amine
N,N-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
3-(furan-2-yl)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
2-cyclopropyl-4-phenyl-9-[2-(pyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
6-{[2-(aminomethyl)piperidin-1-yl]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(1-ethylpiperidin-3-yl)methyl]methylamine
3-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
6-[(diethylamino)methyl]-N-(furan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
ethyl 4-(cyclopropylmethyl)-1-(2-methoxyquinoline-4-carbonyl)piperidine-4-carboxylate
7-[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]-4-methyl-1,2-dihydroquinolin-2-one
3-(4-fluorophenyl)-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
1-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carboxamide