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7-methyl-3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}-1,2-dihydroquinolin-2-one
N-benzyl-N-methyl-3-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-[(2-fluoro-5-methylphenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(3S,9aR)-8-(3-chlorobenzoyl)-3-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-(1H-pyrrole-2-carbonyl)-8-azabicyclo[3.2.1]octane
4-(2,4-dimethoxypyrimidin-5-yl)isoquinoline
methyl 5-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(3R,4S)-1-[3-(piperidine-1-carbonyl)pyridin-2-yl]-4-propylpyrrolidin-3-yl]acetamide
1,3-dimethyl-6-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{1-hydroxy-2-[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}phenol
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
1-(furan-2-carbonyl)-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-1,4-diazepane
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
3-{4-[6-amino-5-cyano-4-(2-methoxyphenyl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}propanoic acid
1-benzyl-4-[3-(methoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methyl-1H-1,2,3-triazole
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
1-{2-oxo-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}piperidin-2-one
5-(2H-1,3-benzodioxole-5-carbonyl)-3-(2,5-dimethylfuran-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(1S,5R)-3-cyclobutanecarbonyl-N-[(2-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-cyclopentanecarbonyl-N-(4-fluorophenyl)piperidin-3-amine
3-(2-ethyl-1H-imidazol-1-yl)-1-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}propan-1-one
4-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-2-one
3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[2-(methylsulfanyl)phenyl]methyl}amine
2-[1-butyl-5-(pyrazin-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
1-methyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-3-fluorophenol
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-(1-methyl-1H-indazol-5-yl)-3-({methyl[(3-methyloxetan-3-yl)methyl]amino}methyl)benzamide
1-ethyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-(5-{[4-(3-fluoropyridin-2-yl)piperazin-1-yl]methyl}furan-2-yl)benzonitrile
N-[2-(oxan-2-yl)ethyl]-3-(piperazine-1-sulfonyl)benzamide
N-[2-(4-{6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}phenoxy)ethyl]acetamide
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
1-(3-methylphenyl)-4-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperazine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-1,2-oxazole-3-carboxamide
5-(cyclopentylamino)-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-cyclohexylurea
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
6-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1H-indole-3-carboxamide
1-[2-(benzyloxy)ethyl]-4-(3-hydroxypropyl)-1,4-diazepan-6-ol
8-[(4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]quinoline
5-amino-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-phenyl-1H-pyrazole-3-carboxamide
(3S,4R)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-phenylpyrrolidine-3-carboxylic acid
(3S,4R)-1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid