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(4aS,8aR)-6-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
3-[(2,4-difluorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
N-(2,3-dihydro-1H-inden-5-yl)-2-(4-methanesulfonylmorpholin-3-yl)acetamide
4,6-dimethyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-methylphenyl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
2-methoxy-4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-3-carbonitrile
2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-1,3-benzodiazole
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(prop-2-en-1-yloxy)benzoyl]-decahydro-1,6-naphthyridin-2-one
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
4-[1-(1H-1,2,4-triazol-5-yl)ethyl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
[3-(2-methylpropyl)-1-[2-(morpholine-4-carbonyl)pyridin-4-yl]piperidin-3-yl]methanol
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
N-cyclopropyl-1-(2-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
2-[benzyl(methyl)amino]-N-methyl-N-(1H-pyrazol-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-cyclopentyl-4-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)benzamide
N-cyclopropyl-1-[(1s,4s)-4-{[(3,4-difluorophenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4aR,7aS)-1-acetyl-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2,1,3-benzoxadiazol-5-ylmethyl)[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amine
(2S,4S)-4-cyclobutaneamido-N-ethyl-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]pyrrolidine-2-carboxamide
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(1,2-oxazol-3-ylmethyl)amine
3-({[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)propanamide
N-(1-methyl-1H-imidazol-2-yl)-3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)benzamide
7-cyclopentyl-2-[2-(4H-1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(2E)-3-(3-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]prop-2-en-1-one
1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
9-(3-hydroxybenzoyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
[(2-chloro-5-fluorophenyl)methyl](ethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
ethyl 4-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]piperidine-1-carboxylate
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]phenyl}acetamide
4-{1-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}pyridine
2-(1-{[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-4-methylpyrimidine-5-carboxamide
1-[3-(2-{3-[(dimethylamino)methyl]phenyl}-1H-imidazol-1-yl)phenyl]ethan-1-one
5-acetyl-3-[1-butyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
methyl 5-[(8-methoxy-2H-chromen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(pyridin-3-yl)acetamide
2-methyl-5-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine
1-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]phenyl}-1H-1,2,4-triazole
(3S,5S)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
N-(1-benzylpyrrolidin-3-yl)-3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)propanamide
3-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(1-methyl-1H-indazol-6-yl)urea
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-phenoxypropan-1-one