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2-{4-[2-(2,3,6-trimethylphenoxy)acetyl]morpholin-3-yl}acetic acid
2-(4-fluorophenoxy)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]acetamide
2-(2-chlorophenyl)-2-hydroxy-1-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]ethan-1-one
1-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-4-phenylpyrrolidin-2-one
(1R,5S)-6-{5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}-6-azabicyclo[3.2.1]octane
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-{[4-(hydroxymethyl)phenyl]methyl}urea
2-(4-methoxy-3,5-dimethylbenzoyl)-1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
1'-(4-methoxypyrimidin-2-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-(1-methyl-1H-pyrazol-4-yl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-{[(3-fluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[1-(3-cyanopyridin-2-yl)piperidin-3-yl]methyl}-4-phenylbenzamide
1-[2-(dimethylamino)acetyl]-4-(4-fluorophenoxy)piperidine-4-carboxylic acid
1-{4-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
4-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)benzonitrile
1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(thiophen-3-yl)propan-1-one
ethyl 2-[4-({[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamoyl}amino)phenyl]acetate
1-cyclopentyl-4-({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)piperazin-2-one
4-cyano-1-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-pyrrole-2-carboxamide
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(3-fluorophenyl)propan-1-one
1-{4-[3-({[(2,4,5-trimethylphenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
2-(4-{[2-(furan-2-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
1-[2-(2-chlorophenyl)ethyl]-2-(propan-2-yl)-1H-imidazole
2-amino-6-{4-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
2-[1-(phenoxymethyl)cyclopropyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(5-methylpyrazin-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
7-(3-methoxyphenyl)-2-(5-methyl-1,2,4-oxadiazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{4-[(4-acetylpiperazin-1-yl)methyl]phenyl}-6-butyl-3,4-dihydropyrimidin-4-one
7-(2-methoxyethyl)-2-(4-propylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-2-yl]-1,3-thiazole
3-(2-methoxyphenyl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
8-methyl-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(pyrimidin-5-yl)quinoline
5-ethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
8-chloro-2-[(cyclobutylamino)methyl]quinolin-4-ol
1-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2,3-dihydro-1-benzofuran-5-carboxamide
5-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
3,4-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
{4-[5-(oxolan-2-yl)thiophene-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
5-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}-2-methoxypyridine
(1R,3S)-3-(2-hydroxyethoxy)-7-(4-methyl-1,3-thiazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
N-[2-(2-chlorophenyl)-1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
3-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
(2S)-2-hydroxy-4-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]butanoic acid
5-[1-(3,4-difluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1-methyl-1H-pyrrole-3-carbonitrile