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4-[(4-{2-[1-(pyridine-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine-1-carbaldehyde
(1S,9aR)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-octahydro-1H-quinolizine
1-(2-methoxyphenyl)-4-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)piperazine
(3S,4R)-1-(6-methylpyridine-3-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}-N-(4-fluoro-2-methylphenyl)propanamide
4-{4-[(5-methoxy-1H-indazol-3-yl)methyl]piperazin-1-yl}quinazoline
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
2-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-3-ol
(4-fluoro-7-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
8-(2-propylpyridine-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-aminopyrimidin-2-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
4-{3-carbamoyl-5H,6H,7H-cyclopenta[b]pyridin-2-yl}-1-methylpiperazine-2-carboxylic acid
1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-ol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(4-cyclopentylphenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid
4-ethyl-3-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(piperidin-1-yl)acetamide
1-[2-(4-chlorophenyl)ethyl]-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-oxopiperidine-3-carboxamide
N4-[2-(quinolin-8-yloxy)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-ethyl-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[4-(2,4-dimethylquinoline-7-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-[(2-chlorophenyl)methyl]-4-[3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-(piperidin-1-yl)-2-[4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]ethan-1-one
N3-[1-(4-chlorophenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-1,4-dihydropyridin-4-one
8-[3-(benzyloxy)propyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
[5-(3-methyl-3-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-2-yl]methanol
1-methyl-N-[2-(2-methyl-1H-indol-3-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
2-(1-{[1-(furan-3-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
ethyl 1-(2,6-dimethoxypyridine-3-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl](1,3-thiazol-4-ylmethyl)amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[2-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)phenyl]-N-methylthiophene-2-carboxamide
9-(1,3-benzothiazol-2-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methanesulfonamide
(4aS,8aR)-6-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
1-(4-fluorophenyl)-4-{[5-(oxan-2-yl)furan-2-yl]methyl}-1,4-diazepane
(2S,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-(1H-pyrazol-5-ylmethyl)pyrrolidine-2-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2,2-dimethyl-1-(thiophen-2-yl)cyclopropane-1-carboxamide
9-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-[(4-chlorophenyl)methyl]-6-oxo-N-(3-phenylpropyl)piperidine-3-carboxamide
N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
2-(1-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-(quinolin-2-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate