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N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
5-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(2-methylphenyl)-1,2,4-oxadiazole
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(1H-pyrrole-3-carbonyl)piperidine
1-[(2,3-dichloro-6-fluorophenyl)methyl]-3-methylpyrrolidin-2-one
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
1-[2-(4-methoxyphenyl)ethyl]-5-[(3-methoxyphenyl)methyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
5-[6-amino-5-cyano-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
N-benzyl-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpiperidin-3-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](pyridin-4-ylmethyl)amine
1-{3-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3-oxopropyl}azepan-2-one
1-[3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
1-ethyl-4,6-dimethyl-2-oxo-N-[3-(3-oxopiperazin-1-yl)propyl]-1,2-dihydropyridine-3-carboxamide
4-(hydroxymethyl)-1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidin-4-ol
1-(furan-2-ylmethyl)-N-(2-hydroxy-3-phenoxypropyl)piperidine-4-carboxamide
3-{5-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-(4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
[(1S)-1-[3-cyclopropyl-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-phenylethyl]dimethylamine
4-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N'-(2-fluoro-5-methylphenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]butanediamide
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N-ethyl-N-(2-hydroxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)methyl]piperidin-3-ol
4-(3-amino-1H-1,2,4-triazole-5-carbonyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
2-{methyl[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethan-1-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
4-fluoro-3-{3-methyl-5-[(2-oxo-1,3-oxazolidin-3-yl)methyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
N-benzyl-5-(1H-indol-2-ylmethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-chloro-5-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydropyridin-2-one
1-(furan-2-ylmethyl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidine-3-carboxamide
1-(1-cyclopentylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2-fluorophenyl)-2-[5-methyl-4-(4-phenylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
2-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-2-(thiophen-2-ylformamido)propanamide
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
4-chloro-1-ethyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
{2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}urea
3-(5-methyl-1,2,4-oxadiazol-3-yl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine
6-methoxy-3-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
6-{1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]piperidin-4-yl}-2-methylpyrimidin-4-ol
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-methylpentane-1,2-dione
N-({1-[(1,4-dimethylpiperidin-4-yl)methyl]piperidin-3-yl}methyl)thiophene-3-carboxamide
N-cyclopropyl-4-methoxy-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-({4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}methyl)piperidine
1-(1-benzyl-1H-pyrazole-4-carbonyl)-1,2,3,6-tetrahydropyridine
2-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-cyclopropyl-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-[3-(4-methylpiperazin-1-yl)butyl]-2-[(prop-2-en-1-yl)amino]benzamide