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(1S,5R)-6-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine
1-methyl-4-[3-(pyridin-2-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{[6-(2,3-dichlorophenyl)pyrimidin-4-yl]amino}ethan-1-ol
N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-sulfonamide
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)-N-propylpropanamide
ethyl 1-{3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidine-2-carboxylate
propan-2-yl 3-{[2-(aminomethyl)piperidine-1-carbonyl]amino}-4-chlorobenzoate
2-fluoro-4-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
(1S,5R)-N-(3-fluorophenyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(dimethylamino)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
(1R,9aR)-1-({[2-(4-methylbenzenesulfonyl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4,6-dimethyl-2-oxo-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carboxamide
N'-cycloheptyl-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}butanediamide
(3S)-3-benzyl-4-(2,3-dimethylquinoxaline-6-carbonyl)piperazin-2-one
1-methyl-4-{5-[4-(trifluoromethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}piperidine
6-cyano-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]pyridine-3-carboxamide
N2-[(4-methanesulfonylmorpholin-2-yl)methyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
3-[5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-{2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-3,3-dimethylurea
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
1-(1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole-5-carboxamide
1-[3-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)-2,4,6-trimethylphenyl]ethan-1-one
(1,3-benzoxazol-2-ylmethyl)({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl})methylamine
N-(2,3-dihydro-1H-inden-2-yl)-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N,2-dimethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}thieno[3,2-d]pyrimidin-4-amine
4-phenyl-1-[(4-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperidine
2-(2H-1,3-benzodioxol-5-yl)-1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
1-{imidazo[1,2-a]pyridine-3-carbonyl}-3-(1H-pyrazol-5-yl)piperidine
N-(3-methoxypropyl)-N-[(4-methylphenyl)methyl]-2-(1H-pyrazol-1-yl)acetamide
(3R,4R)-4-(azepan-1-yl)-1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-ol
3-(propan-2-yl)-5-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,2-oxazole
4-methyl-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-imidazole
N-[1-(thian-4-yl)piperidin-4-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-ethyl-5-{[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl 2-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]sulfonyl}benzoate
2-({2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}amino)pyridine-4-carboxamide
2-cyclopropyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,4-dimethylpyrimidine-5-carboxamide
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methoxyphenyl)-2-methylpiperazine
5-methyl-N-[(1r,4r)-4-hydroxycyclohexyl]-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-(2-methoxyphenyl)-5-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
N-cyclopropyl-4-{[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]amino}pyridine-2-carboxamide
3-(1-oxo-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-2-yl)-3,4-dihydroquinazolin-4-one
1-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}-2-(pyridin-3-yl)ethane-1,2-dione
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide