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1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
(3-{[1-(3,4-dimethoxybenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-(1-benzoxepine-4-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-(2-methoxyacetyl)-N-methyl-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(3S,4R)-1-(2-amino-2-methylpropanoyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
8-(3-hydroxypropanoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(adamantan-1-yl)-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-3-(pyridin-3-yl)propanamide
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-N-(thiophen-2-ylmethyl)pyrimidin-2-amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)benzamide
3-benzyl-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(5-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]dimethylamine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]propanamide
(4aS,8aR)-6-(furan-3-ylmethyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-cyclobutanecarbonyl-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
1-(cyclopropylmethyl)-5-[(1-methyl-1H-indol-3-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
benzyl (7R,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[3-(methylsulfanyl)propyl](pyridin-4-ylmethyl)amine
ethyl 1-({3-[(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)piperidine-2-carboxylate
N-methyl-N-(1H-pyrazol-5-ylmethyl)-2,3-dihydro-1-benzofuran-7-carboxamide
2-amino-5-methyl-6-(5-methylfuran-2-yl)-4-(pyridin-4-yl)pyridine-3-carbonitrile
2-(3-fluorophenoxymethyl)-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
(2R)-2-acetamido-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}propanamide
(2-{4-[1-(dimethylamino)ethyl]phenyl}pyridin-4-yl)methanol
(4aR,7aS)-1-(2-hydroxyethyl)-4-(4-methoxy-2-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(2-oxoazepan-1-yl)propanamide
1-(1-methyl-1H-1,3-benzodiazol-2-yl)ethane-1,2-diol
(2-{4-[2-chloro-5-(trifluoromethyl)benzoyl]morpholin-2-yl}ethyl)dimethylamine
2-[2-chloro-4-(7-methoxy-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)phenoxy]acetamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-(2-hydroxyethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-4-(1H-pyrazol-1-yl)benzamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
4-[4-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)phenyl]but-3-yn-1-ol
5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-(2-methoxyethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazole
(2S,6S)-1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-(3-ethylphenyl)-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[(2,3,4-trifluorophenyl)carbamoyl]methyl}propanamide
methyl 2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyridine-3-carboxylate
3-(1-{[1-(2-methylpyridin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propanoic acid
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxylic acid
1-[(2-methoxy-4-methylphenyl)methyl]-4-(methoxymethyl)piperidine
1-benzyl-N,N-dimethyl-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-(4-methoxyphenyl)-1H-indazole
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,N-dimethylpyrimidin-4-amine
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-(phenylsulfanyl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
N-cyclopropyl-6-methoxy-3-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-2-carboxamide
2-[(3,4-dimethoxyphenyl)methyl]-N-(2-hydroxypropyl)-N-methyl-1,3-benzoxazole-6-carboxamide