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N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
3-(2-methylphenyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
N-[(3R,4R)-3-hydroxy-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl]pyrazine-2-carboxamide
2-(ethanesulfonyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1-(2-phenylethyl)-1H-imidazole
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2,8-dimethylquinoline
3-{[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
3-(5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
3-[1-(6-cyanopyridin-2-yl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-1,2,3,6-tetrahydropyridine
6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-2-one
ethyl 3-benzyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine-3-carboxylate
N-methyl-2-(1H-pyrazol-1-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
1-{2-[1-(3-methylpyridin-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
1-methyl-4-(1-{1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl}ethyl)piperazine
(2S,4S)-4-amino-N,N-diethyl-1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidine-2-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]pyrrolidin-3-yl]acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carboxamide
1-(adamantan-1-yl)-4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazine
7-(1,3-benzothiazol-2-yl)-4-[(2-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,6R)-9-{[3-methoxy-4-(pyrrolidin-1-yl)phenyl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
4,5-dimethyl-6-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidine
8-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1-oxa-8-azaspiro[4.6]undecane
4-[(2-methylpyrrolidin-1-yl)methyl]-N-(1-propyl-1H-1,2,4-triazol-3-yl)benzamide
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
2-methyl-3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyridin-2-amine
2,2-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}oxane-4-carboxamide
2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinolin-4-ol
4-(1-ethyl-1H-imidazol-2-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine
3-[1-(1-ethylpiperidine-2-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
7-fluoro-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[(3-methylpyridin-2-yl)methyl]quinoline-4-carboxamide
1-(1,3-dihydroxypropan-2-yl)-4-[3-(1H-pyrazol-4-yl)propanoyl]-1,4-diazepane-6-carboxylic acid
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-N-benzylpyrimidin-2-amine
N-{2-[methyl(2-phenylethyl)amino]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(1,2-benzoxazol-3-yl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}acetamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]pentan-1-one
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){1-[1-(5-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-2-phenylethyl}amine
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-chlorophenyl)-N-methyl-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
3-fluoro-4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
4-[2-methyl-4-(3-methylphenyl)-5-oxopiperazine-1-carbonyl]benzonitrile
[2,4,6-trimethyl-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenyl]methanol
3-{2-[(1R,5S)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
5-[2-(benzenesulfonyl)ethyl]-1-ethyl-1H-1,2,4-triazole
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(5-ethylpyridin-2-yl)methyl]amine
1-(3-fluoropyridin-4-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide