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3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(2-chloro-6-methylphenyl)urea
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
N-[furan-2-yl(phenyl)methyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
1-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazine
2-(3-aminopyrrolidine-1-carbonyl)-6-(4-methoxyphenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(4-cyclopentylpiperazin-1-yl)-2-(dimethylamino)-2-(4-fluorophenyl)ethan-1-one
5-methyl-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,3-oxazole
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-cyclohexyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
{1-[5-(2-chlorophenyl)-2-methylfuran-3-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
2-(2H-indazol-2-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
1-(3,5-dimethylbenzoyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
5-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}pyridine-2-carbonitrile
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
3-(diphenylmethyl)-N-(5-hydroxyadamantan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}propan-1-one
3-(1H-1,3-benzodiazol-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[3-(1H-indazol-1-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-{[3-(pyridin-2-yl)phenyl]methyl}-2-(trifluoromethyl)morpholine
N-cyclopropyl-3-{5-[5-(methoxymethyl)furan-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[3-(3,4-dimethoxyphenyl)propyl]-3-(1,2-oxazinan-2-yl)propanamide
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
2-(3-methoxyphenoxymethyl)-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
5-methyl-4-{[2-(1H-1,2,4-triazol-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-4-phenylazepane-1-carboxamide
N-(2-oxoazepan-3-yl)-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
2-{1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-5-fluoro-1H-1,3-benzodiazole
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
6-(2-hydroxyethyl)-N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
[(1-cyclohexylpiperidin-3-yl)methyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-3-ylmethyl)amine
4-(5-ethylfuran-2-yl)-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole
4-(5-fluoro-2-methylphenyl)-3-(1H-pyrazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[2-(methoxymethyl)piperidin-1-yl]ethan-1-one
ethyl 1-[(3-chloro-4-hydroxyphenyl)methyl]-4-(cyclopropylmethyl)piperidine-4-carboxylate
N-(3-{4-[(2-methoxyethyl)amino]piperidin-1-yl}phenyl)-4-phenylbutanamide
1-methyl-2-(morpholin-4-yl)-5-(3-propyl-1,2,4-oxadiazol-5-yl)-1H-1,3-benzodiazole
4-chloro-2-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
6-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-2-methylpyrimidin-4-ol
2-[3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4H-chromen-4-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[2-(3-methylphenoxy)acetyl]-1-(4-methylphenyl)piperazin-2-one
N-methyl-N-{1-[2-(2-oxo-1,2-dihydroquinolin-1-yl)acetyl]pyrrolidin-3-yl}acetamide
5-benzenesulfonamido-1-ethyl-N,2-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[2-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
N-benzyl-N,1-dimethyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-{[4-(dimethylamino)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate