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4-(5-{[4-(1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(1R,5R)-6-benzyl-3-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2-aminoethyl)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-1,2,3-triazole-4-carboxamide
N4-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N1,N1-dimethylpiperidine-1,4-dicarboxamide
5-methyl-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(6-hydroxy-1,4-diazepane-1-carbonyl)-1,2,3,4-tetrahydroquinoxalin-2-one
1-(3-methoxyphenyl)-2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethan-1-ol
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
4-benzyl-1-(1H-imidazol-4-ylmethyl)piperidine-4-carboxylic acid
3-benzyl-5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-yl]-1H-1,2,4-triazole
8-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-cyclobutyl-5-(trifluoromethyl)-1H-1,3-benzodiazole
4-{1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]piperidin-3-yl}benzoic acid
3-(butan-2-yl)-1-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]urea
(1R,5S)-3-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-yl]acetamide
5-(furan-2-yl)-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-1H-imidazole
4-benzyl-N,3-diethyl-5-oxo-1,4-diazepane-1-carboxamide
1-cyclohexyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidine-4-carboxamide
2-{5-[1-(difluoromethyl)-1H-pyrazol-3-yl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(methylamino)ethyl]amine
1-(2-chloropyridin-3-yl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
3-(2-methylquinolin-5-yl)pyrazine-2-carbonitrile
2,6-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]quinoline-4-carboxamide
2-[(6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-yl)amino]ethan-1-ol
N-[1-(1-propylpiperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
3-{1-[1-(1-cyclopropylpropan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
3-hydroxy-3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-1-(3-phenylpropyl)piperidin-2-one
methyl 6-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrimidine-4-carboxylate
N4-methyl-N4-[2-(morpholin-4-yl)propyl]-6-(propan-2-yloxy)pyrimidine-2,4-diamine
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-3-fluoro-N-(2-methoxyethyl)benzamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-({5-[1-(3,3-dimethylbutyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[(3S)-3-ethylmorpholine-4-carbonyl]-N-methyl-1,3-thiazol-2-amine
4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(pyridin-3-yl)morpholine
2-[4-(4,6-dimethoxypyrimidin-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-methyl-8-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
1-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
(1R,6S)-3-(3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonyl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane
2-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
3-[2-(2,6-difluorophenyl)ethyl]-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
1-[(4-fluorophenyl)methyl]-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole