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4-(3-benzyl-1H-pyrazol-5-yl)-1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
2-amino-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(2S,4R)-1-(1H-imidazol-4-ylmethyl)-N-(propan-2-yl)-4-[2-(propylsulfanyl)acetamido]pyrrolidine-2-carboxamide
3-(5-fluoropyridin-3-yl)-1-[2-(4-methoxyphenyl)ethyl]-1-(oxolan-2-ylmethyl)urea
N-[4-methoxy-3-({[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)phenyl]acetamide
2-(2,4-difluorophenoxy)-1-(6-methyl-2-phenyl-1,2-diazinan-1-yl)ethan-1-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-phenylmethanesulfonylpiperidine
2-{9-[(2-fluorophenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-[4-(3-fluorophenyl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylcyclopentanecarbonyl)piperidine
8-[(2S,3R)-2-amino-3-hydroxybutanoyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(1H-indol-1-ylmethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
1-[5-({[(2-chlorophenyl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
4-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
3-(1H-imidazol-2-yl)-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-ol
5-{2-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrimidin-2-amine
2-(4-chlorophenyl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazole
N-[(1-benzylpyrrolidin-3-yl)methyl]-N-methylpyrimidin-4-amine
4-[4-(1-methoxypropan-2-yl)piperidin-1-yl]-2-methyl-6-(piperidin-4-yl)pyrimidine
6-(2-aminoethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methylpyrimidin-4-amine
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl][(8-methoxyquinolin-2-yl)methyl]methylamine
4-(1-phenyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-2-amine
4-(2-methoxypyridin-3-yl)-6-methyl-1,3-benzothiazol-2-amine
[1-(oxane-4-carbonyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
N-(1-cyclopentyl-1H-pyrazol-5-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
4-(1-{4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl}ethyl)morpholine
5-(4-aminopiperidine-1-carbonyl)-2-(3,5-dichlorophenyl)pyrimidin-4-ol
1-(4-{4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2-methoxyphenoxy}piperidin-1-yl)ethan-1-one
4-chloro-1-methyl-3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}-1H-indazole
4-(furan-3-ylmethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
2-{2-[(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)formamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
7-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
1-(azepan-1-yl)-3-(3-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}phenoxy)propan-2-ol
3-ethyl-5-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
3-[(3-ethenylphenyl)methyl]-9-(furan-2-carbonyl)-3,9-diazaspiro[5.5]undecane
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(4-fluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[4-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
3-{[1-(4-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-[(5-fluoro-2-methylphenyl)methyl]-4-(2,3,5-trifluorophenyl)-1H-1,2,3-triazole
1-{3-[3-(2-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(propan-2-yl)-3-(1H-pyrazol-1-yl)benzamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-sulfonamide
1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
ethyl 1-[(3-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate