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2-{6-hydroxy-4-[3-(1H-imidazol-2-yl)benzoyl]-1,4-diazepan-1-yl}acetic acid
(4aS,8aR)-1-(3-aminopropyl)-6-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
5-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}-N-propylpyrimidin-2-amine
ethyl 1-[(2-hydroxy-3-methoxyphenyl)methyl]-3-(2-phenylethyl)piperidine-3-carboxylate
7-(2-hydroxyethyl)-2-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[5-(2-chloro-6-fluoro-3-methylphenyl)-1,2,4-oxadiazol-3-yl]pyridazine
1-(2,4-dimethylpyrimidine-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-ethyl-5-methyl-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-2-yl)pyridine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(4-methoxyphenyl)acetamide
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1H-pyrazole-4-carboxamide
4-(2-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)phenol
[2-(2-chloro-6-methylphenoxy)ethyl]({[3-(morpholin-4-ylmethyl)phenyl]methyl})amine
(1s,4s)-4-{4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
(2S,4R)-N-(propan-2-yl)-4-{4-[(N,3,3-trimethylbutanamido)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
1-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
8-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-1-oxa-8-azaspiro[4.5]decane
(3S)-1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-amine
ethyl 2-{1-[6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-amido]cyclohexyl}acetate
methyl[(3-methyl-1H-indol-2-yl)methyl][(1-methylpiperidin-2-yl)methyl]amine
2-{[5-(1H-imidazol-1-ylmethyl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-[4-(4-cyclopentylpyrimidin-2-yl)piperazin-1-yl]propan-1-ol
(3S,9aR)-3-benzyl-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-fluoro-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}pyridazine
1-ethyl-5-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-[4-(4-fluorophenyl)oxane-4-carbonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
2-[(3-chlorophenyl)methyl]-6-[3-(methoxymethyl)piperidine-1-carbonyl]-1,3-benzoxazole
3-[(3R,4S)-1-(2-methylpyrimidin-4-yl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-(1H-imidazol-1-ylmethyl)-1-(4,4,4-trifluorobutyl)piperidine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
5-{[(2-methoxyphenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 2-chloro-5-{[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]amino}benzoate
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(4-methyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(4-methylpiperazin-1-yl)propanamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
4-(5-ethyl-2-methylpyrimidin-4-yl)-2-(4-fluorophenyl)morpholine
6-[3-(morpholin-4-ylmethyl)phenyl]quinolin-4-amine
1-ethyl-4,6-dimethyl-2-oxo-N-{1-[2-(trifluoromethyl)phenyl]ethyl}-1,2-dihydropyridine-3-carboxamide
3-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanoic acid
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]ethan-1-one
(1R,3S)-7-[4-methyl-6-(methylamino)pyrimidin-2-yl]-7-azaspiro[3.5]nonane-1,3-diol
N-cyclohexyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(thiophen-3-ylmethyl)acetamide
3-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N,N-dimethylpyrazin-2-amine
7-(cyclopropylmethyl)-2-(8-methoxyquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(3aR,6aS)-5-[2-(azepan-1-yl)acetyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide