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(2R)-2-hydroxy-3-methyl-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-one
N-(2,3-dihydroxypropyl)-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-methyl-2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(1,3-dimethyl-1H-pyrazol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(dimethylsulfamoyl)-N-[4-(3-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
3-{2-oxo-2-[3-(pyridin-2-yl)azetidin-1-yl]ethyl}imidazolidine-2,4-dione
4-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}-2,1,3-benzoxadiazole
dimethyl[1-(3-{1-[(5-methylpyrazin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]amine
2-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
4-{2-[1-(quinoxaline-6-carbonyl)piperidin-2-yl]ethyl}phenol
1-[(2-fluorophenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(3-benzoylpiperidin-1-yl)-2-(2-methoxyphenoxy)ethan-1-one
6-ethyl-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-({4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-3,4-dimethoxypyridine
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-4-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(furan-2-ylmethyl)pyrimidin-2-amine
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-methoxyfuran-2-carbonyl)piperidine
N-ethyl-N-(2-hydroxyethyl)-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(3-methylpyridin-4-yl)-4-[1-(pyrimidin-2-yl)piperidin-4-yl]-1,4-diazepane
2-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,2-oxazinane
3-methanesulfonamido-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)propanamide
4-ethyl-1-[(3-phenoxyphenyl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-hydroxy-4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pentanamide
4-methyl-6-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-5-(prop-2-en-1-yl)pyrimidin-2-amine
N-[3-(azepan-1-yl)propyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(1H-pyrazol-1-yl)butanamide
N-[1-(furan-2-yl)ethyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
1-{[2-(difluoromethoxy)phenyl]methyl}-3-(2-methoxyphenoxy)azetidine
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
N-cyclopropyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(1,3-thiazol-2-ylmethyl)acetamide
3-(3-hydroxy-3-methylbutyl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]benzamide
3-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
2-(3-hydroxyphenyl)-1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]ethan-1-one
methyl 2-{4-[3-(1H-imidazol-1-yl)propyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
3-benzyl-4-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperazin-2-one
5-methoxy-9-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
2-{[(3,5-dimethylphenyl)methyl]sulfanyl}-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
3-(2,6-dimethylphenoxy)-1-(2-fluoro-4-methylbenzoyl)azetidine
N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
(3aS,6aS)-2-acetyl-5-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-4-{[(2,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrrole-2-carboxamide
4-[1-(4-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]pyridazine
1-(furan-2-carbonyl)-4-[(8-methoxy-2H-chromen-3-yl)methyl]-1,4-diazepane
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine