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2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
N-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)benzamide
1-[(2-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}phenyl)methyl]pyrrolidin-2-one
8-(3-ethyl-1,2-oxazole-5-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
4-methyl-6-{4-[1-(2-methylphenyl)piperidin-4-yl]piperazin-1-yl}pyrimidin-2-amine
2-methyl-4-[3-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)phenyl]but-3-yn-2-ol
2-amino-3-ethyl-N-[2-(2-fluorophenoxy)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1S)-1-phenylethyl]urea
1-[(3,4-dimethylphenyl)methyl]-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
5-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-ethylpyrimidin-2-amine
1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-(4-methoxyphenoxymethyl)piperidine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
(2-{[1-(4,6-dimethylquinolin-2-yl)piperidin-4-yl]oxy}ethyl)dimethylamine
(3E)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pent-3-en-1-one
(2S,4S)-4-amino-1-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
6-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
9-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[6-cyclobutanecarbonyl-2-(dimethylamino)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
1-(7-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(propan-2-yloxy)ethan-1-one
methyl (2S,4R)-4-[2-(azocan-1-yl)acetamido]-1-methylpyrrolidine-2-carboxylate
N-[2-(3-methoxyphenyl)-1-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]benzamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-3-(1H-pyrazol-4-yl)benzamide
N-methyl-5-phenyl-N-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
2-{1-[5-(ethanesulfonyl)thiophen-2-yl]-1H-pyrazol-3-yl}pyrazine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(4-methanesulfonylphenyl)methyl]-1H-1,2,4-triazole
5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1H-1,2,3-benzotriazole
N-ethyl-2-[4-(4-methoxybenzoyl)piperazin-1-yl]pyridine-3-carboxamide
3-(2-methylphenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
N-[2-(1,3-benzothiazol-2-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
3-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)-5-(2,3,4-trimethoxyphenyl)benzamide
1-{1'-[(2S)-2-amino-2-phenylacetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
[2-ethoxy-5-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenyl]methanol
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[3-(pyridin-4-yl)propyl]carbamoyl}pyrrolidine-2-carboxylate
3-{3-[3-(quinolin-6-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
3-(2-methylphenyl)-1-[3-(methylsulfanyl)propyl]piperidine
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylacetamide
3-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}-1H-indole
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N,N-bis(2-hydroxyethyl)-2-methyl-1-benzofuran-5-carboxamide
ethyl 1-[(2-chloro-4-hydroxy-5-methoxyphenyl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
1-[(2-fluorophenyl)methyl]-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
3-ethyl-1-[2-(4-ethylpiperazin-1-yl)acetyl]piperidine-3-carboxylic acid