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5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
2-[4-(1,4-dithiepan-6-yl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(pyridin-2-yl)propanamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl){[1-(propan-2-yl)piperidin-4-yl]methyl}amine
4-[1-(cyclopropanesulfonyl)piperidin-3-yl]benzoic acid
methyl 6-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidine-4-carboxylate
(1-{1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
methyl[(4-{2-[1-(4-methylbenzoyl)piperidin-2-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
8-methoxy-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(ethylamino)-4-methyl-N-[1-(pyrazin-2-yl)piperidin-3-yl]-1,3-thiazole-5-carboxamide
1-[(1-methylpiperidin-2-yl)methyl]-1,2-dihydroquinoxalin-2-one
4-methanesulfonyl-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}piperazine-1-carboxamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(2-fluorophenoxy)piperidine
5-ethyl-N-({3-methyl-7-[3-(2-oxopyrrolidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,2-oxazole-3-carboxamide
N-{2-[(1-methoxypropan-2-yl)amino]ethyl}-N-methylmethanesulfonamide
N-[1-(pyrimidin-4-yl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
5-(3,5-dimethyl-1-benzofuran-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
2-methoxy-1-[1'-(1H-1,2,4-triazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
methyl 3-[(4-ethylphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(3-hydroxypropyl)-1-[1-(3-phenylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
8-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(2-{[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]oxy}phenyl)methyl]morpholine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
4-(furan-2-ylmethyl)-3-[hydroxy(phenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl (2S,4S)-4-[2-(2-ethyl-1H-imidazol-1-yl)acetamido]-1-methylpyrrolidine-2-carboxylate
1-(3-methoxypropyl)-8-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methoxy-N-methyl-4-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4H-pyran-2-carboxamide
4-(cyclopropylmethyl)-1-(5-ethylpyrimidin-2-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
1,3-dimethyl-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-pyrazole
N-(2,2-dimethyloxan-4-yl)-N-ethyl-7-fluoro-2-methylquinoline-4-carboxamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
3-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
5-(1-phenylcyclohexanecarbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
N4-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyrimidine-2,4-diamine
N-cyclopropyl-1-{2-[1-(2,5-dimethoxybenzenesulfonyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-hydroxy-3-methylphenyl)methyl]piperidin-3-ol
1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
2-[(3R,4S)-3-(4-chloro-2-methoxybenzamido)-4-cyclopropylpyrrolidin-1-yl]acetic acid
N-cyclopropyl-3-{5-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-1H-indole-6-carboxamide
2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
(1S,5R)-6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[3-(pyridin-3-yl)propyl]benzamide
5-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
3-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-1λ6-thiolane-1,1-dione
2-(2,4-dichlorophenoxy)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
7-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]quinolin-8-ol