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ethyl 2-[4-(2-chlorophenoxy)piperidin-1-yl]-1,3-oxazole-4-carboxylate
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[(3-phenoxyphenyl)methyl]pyrrolidine-2-carboxamide
ethyl 1-benzyl-5-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
1-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine-4-carboxylic acid
5,8-dimethoxy-4-methyl-2-[3-(pyridin-3-yl)azetidin-1-yl]quinoline
2-{4-[(8-methoxyquinolin-2-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
1-[benzyl(methyl)amino]-3-[4-(piperidin-1-ylmethyl)phenoxy]propan-2-ol
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
9-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
5-{4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl}-1-cyclohexyl-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]urea
4-(1,2-oxazolidine-2-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclopent-1-ene-1-carboxamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
(1R,5R)-6-(4-hydroxy-3-methoxybenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
8-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]quinoline
3-(2-ethylbutyl)-8-(quinoline-7-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4S)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
5-(4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenoxymethyl)furan-2-carboxylic acid
2-oxo-8-[2-(pyrrolidin-1-yl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[2-({[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-(2-methylpropyl)piperidin-4-amine
4-[(3-fluorophenyl)methyl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
4-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-{[3-(benzyloxy)phenyl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[methyl(prop-2-yn-1-yl)amino]-2-[4-(propan-2-yloxy)phenyl]acetic acid
8-(5,6-dimethylpyrimidin-4-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(furan-2-yl)propan-1-one
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl](quinolin-2-ylmethyl)amine
3-(2-methoxyphenyl)-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]propan-1-one
8-(3,6-dimethylpyrazin-2-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-1-{[1-(2-methylphenyl)-1H-pyrrol-2-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
[2-(isoquinolin-5-yl)-7-methylquinolin-3-yl]methanol
5-fluoro-1,3-dimethyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
N-methyl-5-[(methylsulfanyl)methyl]-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
2-benzyl-9-[2-(ethylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyridin-4-yl)propyl]pyridin-2-amine
1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-N,N-dimethylpyrrolidin-3-amine
N,N,5-trimethyl-2-{3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-4-amine
(2S,4R)-4-amino-N-ethyl-1-[3-(pyrimidin-2-yloxy)benzoyl]pyrrolidine-2-carboxamide
1-{4-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-1-yl}-3-methylbutan-1-one
N-(4-fluorophenyl)-1-[4-(methylsulfanyl)benzoyl]piperidin-3-amine
4-[({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}amino)methyl]-1-ethylpyrrolidin-2-one