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4-(4-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
methyl 1-[(3S,5S)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(2-methylpropyl)amine
1-[2-(4-fluorophenyl)ethyl]-4-methyl-1,4-diazepan-6-ol
2-[4-(2-cyanobenzoyl)morpholin-3-yl]-N-[3-(pyridin-2-yl)propyl]acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(furan-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-[(4-methylphenyl)sulfanyl]propan-1-one
[(2-fluoro-4-methoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
6-(4-hydroxyphenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-ethyl-5-fluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-2-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(2,5-dimethoxyphenyl)-1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidine
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-[(4aR,7aS)-4-(6-methoxyhexanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
2-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-6-methylphenol
1-(2-ethylbutanoyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
ethyl 1-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-hydroxy-5-(1H-pyrrol-1-yl)benzamide
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
methyl[(5-methylfuran-2-yl)methyl]({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amine
4-{2-[(2-methyl-6-propylpyrimidin-4-yl)oxy]hex-5-en-1-yl}-1,4-oxazepane
3-(1H-1,2,3-benzotriazol-4-yl)-1-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}urea
ethyl 4-(oxan-2-ylmethyl)-1-(3-phenylprop-2-yn-1-yl)piperidine-4-carboxylate
4-[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]piperidine
6-ethyl-N-[furan-2-yl(phenyl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{4-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
1-(2-ethoxyacetyl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-pyrazol-1-ylmethyl)piperidine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]acetamide
6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]but-2-enamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(3-fluoro-4-methoxybenzoyl)piperidine-3-carboxylate
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(piperidin-3-yl)benzamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(oxan-4-yl)piperidine-3-carboxamide
7-chloro-4-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
1-[cyclohexyl(methyl)amino]-3-[3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-(5-methylthiophen-2-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-[2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyridine
(1S,3R)-3-amino-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}cyclopentane-1-carboxamide
2-{1-[3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propyl]piperidin-3-yl}propan-2-ol
4-[(dimethylamino)methyl]-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}azepan-4-ol
[(2-fluoro-4-methoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(3S,9aR)-8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(hydroxymethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,2-dimethyl-4-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
2-[(4-methoxyphenyl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}morpholine
1-(2H-1,3-benzodioxol-5-yl)-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
1-(4-{[(1S,2S)-2-hydroxycyclohexyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one