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2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}acetamide
4-benzoyl-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-(2-phenoxyethyl)propanamide
1-(5-methoxy-2-{[methyl(thian-4-yl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-(4-hydroxypiperidin-1-yl)propan-1-one
5-(5-aminopentyl)-11,13-dimethyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
2-(3-methoxypropyl)-8-{[4-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-benzyl-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,1-dimethyl-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
4-benzyl-1-methyl-3-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
3-hydroxy-3-({[(3-methoxyphenyl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-[(3E)-4-methylhex-3-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
1-[1-(morpholine-4-carbonyl)piperidin-4-yl]-3-(2,3,5-trifluorophenyl)urea
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
7-(propan-2-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
diethyl({[3-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
9-[(2R)-2-hydroxy-3-methylbutanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1,2,5-trimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrrole-3-carboxamide
1-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
methyl 5-[(furan-2-ylmethyl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3-fluorophenyl)methyl]-N-methyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4,6-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(3-methylbutyl)-8-[2-(oxolan-2-ylmethoxy)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(furan-3-ylmethyl)-7-(1H-imidazol-4-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(4-fluorophenyl)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
1-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(1H-imidazol-4-yl)-1H-imidazole
[(2-fluoro-5-methoxyphenyl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-[2-(4-chlorophenyl)-2-hydroxyethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
6-(2,2-dimethylmorpholin-4-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-ethyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-(3,5-dimethylphenyl)-4-(2-ethylpyridine-4-carbonyl)piperazin-2-one
methyl 1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carbonyl]piperidine-2-carboxylate
2,7,8-trimethyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]quinoline-4-carboxamide
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methylimidazolidin-2-one
2-amino-6-{4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)[(2,4,6-trimethoxyphenyl)methyl]amine
4-(3,4-diethoxyphenyl)-2-(1H-imidazol-2-yl)-1H-imidazole
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-ethyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N4-[2-(2-ethoxyethoxy)phenyl]-N1,N1-dimethylpiperazine-1,4-dicarboxamide
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-4-(pyridin-4-yl)pyrimidin-2-amine
1-ethyl-4-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[2-(dimethylamino)ethyl]-9-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
2-(2-{[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1S,5R)-6-methyl-3-[2-(4-phenylphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one