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1-(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-3-phenylpropan-1-ol
2-methoxy-2-methyl-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]acetamide
N5-[2-(2-fluorophenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(2-methoxyphenyl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}propan-1-one
methyl 6-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}pyridine-2-carboxylate
9-hydroxy-3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}quinoxaline-5-carboxamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-4-(piperidin-1-yl)butanamide
N-(2-methoxyethyl)-3-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)propanamide
ethyl 1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidine-2-carboxylate
(2R,3R,6R)-5-(1-ethyl-1H-pyrazole-5-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-ethyl-1,5-dimethyl-3-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{2-[3-(3-methylphenoxy)azetidin-1-yl]-2-oxoethyl}azepan-2-one
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-(5-methylfuran-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4-(4-chlorophenyl)-3-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazole
2-(cyclopropylmethyl)-9-(2-ethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-oxoethoxy}acetamide
2-methoxy-3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-({1-[6-(1H-indol-3-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-cyclopentyl-2-({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}amino)propanamide
5-methoxy-2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
N-cyclohexyl-3-[(2-methyl-4-phenylpyridin-3-yl)formamido]propanamide
2-ethyl-5-{3-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}pyrimidine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5,6-trimethylpyrimidin-4-amine
3-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)propanamide
3-methyl-1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
N-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
5-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
N6-[1-(3,5-difluorophenyl)ethyl]-N4,N4-dimethylpyrimidine-4,6-diamine
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentan-1-one
6-(4-fluorophenyl)-2-[4-(piperidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(1H-pyrazol-1-yl)acetamide
1-{3-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-(3-methyl-1H-pyrazol-1-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
4-[(4-fluorophenyl)methyl]-1-[2-oxo-2-(piperidin-1-yl)ethyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{3-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
1-{2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]ethyl}piperidin-4-ol
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-(oxolan-2-ylmethyl)-N-propylpiperidin-4-amine
4-(8-methoxyquinolin-5-yl)pyridin-3-amine
5-methyl-4-[3-methyl-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(prop-2-en-1-yl)-1H-pyrazole
3-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-methoxyacetamide
N-ethyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(4aS,7aR)-1-(1-methyl-1H-pyrazole-3-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-1-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-2-methylpropan-1-one
1-(2-methylphenyl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
3-(1-{[1-(2-methoxybenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
1-ethyl-4-{2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carbonyl}piperazin-2-one
5-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine