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2-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidin-1-yl}pyridine-3-carboxamide
2-(4-propanoylphenoxy)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]acetamide
N'-(2-methoxyethyl)-N-(2-methylphenyl)-N'-(3-phenylprop-2-yn-1-yl)propanediamide
4-cyclopropyl-6-[4-(trifluoromethyl)piperidin-1-yl]pyrimidine
1-(4-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N2-benzyl-6-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-1,3,5-triazine-2,4-diamine
4-[3-(5-methylfuran-2-yl)benzoyl]-1λ6-thiomorpholine-1,1-dione
(2S)-2-hydroxy-4-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}butanoic acid
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(1H-pyrazol-3-ylmethyl)-1,4-diazepan-6-yl]oxy}acetamide
3-(4-aminopyrimidin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
2-[4-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)piperazin-1-yl]benzonitrile
1-(4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
1-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]azepan-2-one
1-(3-methylpyridin-2-yl)-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
4-{furo[3,2-c]pyridin-4-yl}-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
(2S,4S)-4-amino-1-(2-ethoxypyridine-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
8-(3-phenylpropyl)-2-(pyridin-3-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]quinoline
N,N-dimethyl-1-{[3-(methylsulfanyl)phenyl]methyl}azepan-4-amine
1-{1-[(2-ethyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
ethyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl](pyridin-4-ylmethyl)amine
2-(1-tert-butyl-1H-pyrazol-4-yl)-4-(2-methylpiperidine-1-carbonyl)quinoline
2-{4-[(5-chlorothiophen-2-yl)methyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
N-methyl-4-(pyrrolidine-1-carbonyl)-6-(3,3,3-trifluoro-2-methylpropyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-methyl-N-(oxan-2-ylmethyl)-3-pentanamidobenzamide
2-[2-(2-methoxyethoxy)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-fluoro-2-methylphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-{1-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}methanesulfonamide
1'-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
(3aS,6aR)-5-benzyl-3-cyclopentyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(2-hydroxyethyl)-4-methoxy-N-methyl-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-methylurea
(1R,3S)-7-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-(oxane-4-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzene-1,3-diol
(2R)-3-(benzyloxy)-2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-1-ol
methyl (2S)-1-[2-(cyclopentylmethyl)-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxylate
5-[2-(2-chlorophenyl)acetyl]-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)pyrrolidin-2-one
4-(2-acetyl-5-methoxyphenoxy)thiane-4-carboxylic acid
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
(2S,4S)-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
6-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-2-carboxylic acid
methyl[(3-{[1-(naphthalene-1-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](quinolin-5-ylmethyl)amine
N-methyl-1-phenyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
3-(2-phenylethyl)-5-(1H-1,2,4-triazol-1-ylmethyl)-1,2,4-oxadiazole