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3-(3-methylbut-2-en-1-yl)-5-(3-phenylpropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-[(6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}pyrimidin-4-yl)amino]ethan-1-ol
3-[(2-methoxynaphthalen-1-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
3-{2-[methyl({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-[(3-chlorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(dimethylamino)-2-(4-methylphenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
2-ethyl-5-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]pyrimidine
2-[(4-benzoylpiperazin-1-yl)methyl]-3-methoxyphenol
N1-[4-(trifluoromethyl)pyridin-2-yl]ethane-1,2-diamine
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-cyclopropanecarbonyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-4-carboxamide
4,4,4-trifluoro-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}butanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]pyrrolidine-1-sulfonamide
2-{4-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
1-cyclopentyl-3-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidine
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-hydroxy-2-methylpropan-2-yl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-{4-[1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-3-methylurea
1-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
1'-[4-(morpholin-4-yl)benzoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
3-{[(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]methyl}piperidin-3-ol
3-hydroxy-3-({[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
methyl 2-(azocane-1-sulfonyl)-6-cyclohexanecarbonyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(4-cyclopentyl-1,4-diazepan-1-yl)-3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropan-1-one
4-[4-(2-fluorophenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-(3-{2-[(dimethylcarbamoyl)amino]acetamido}phenyl)-4-methylbenzamide
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-methyl-7-{2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl (2S)-1-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidine-2-carboxylate
1-ethyl-5-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(1-{1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-[(methylsulfanyl)methyl]piperidine
(3E)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]hept-3-enoic acid
4-[(4-fluorophenyl)methyl]-1-(furan-2-ylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
[(2S,4R)-4-(dimethylamino)-1-({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-2-yl]methanol
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(4-cyclopentylpiperazin-1-yl)-N-ethyl-N-phenylpropanamide
5-propyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-1-cyclopentylpiperazin-2-one
N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-2,3-dimethyl-1H-indole-7-carboxamide
2-{4-[(3-methylfuran-2-yl)methyl]piperazin-1-yl}pyrimidine
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
methyl (1R,3S,3aR,6aS)-1-benzyl-5-methyl-4,6-dioxo-3-(1,2,3-thiadiazol-4-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
ethyl 2-{1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]piperidin-2-yl}acetate
N-cyclopropyl-3-{5-[(2-methyl-1-benzothiophen-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[2-(dimethylamino)ethyl]-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide