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6-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
5-[(4-acetyl-1,4-diazepan-1-yl)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
7-(2,3-dihydro-1H-inden-2-yl)-2-oxa-7-azaspiro[4.5]decan-8-one
7-(cyclohexylmethyl)-2-ethyl-2,7-diazaspiro[4.5]decan-6-one
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
(3S,4R)-3-acetamido-4-(4-methoxyphenyl)-N-(2-phenylethyl)pyrrolidine-1-carboxamide
2-methyl-8-(1-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
N-{1-[7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}methanesulfonamide
7-(3-chlorophenyl)-4-[3-(dimethylamino)pyrazin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{3-[2-(2-hydroxyethyl)-4-methyl-1H-1,3-benzodiazol-1-yl]phenyl}-2-methoxyacetamide
3-methyl-4-[3-phenyl-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazol-1-yl]pyridine
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-{[(4aS,8aR)-4a-(hydroxymethyl)-6-propyl-decahydro-1,6-naphthyridin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
(3aS,6aS)-2-cyclopentyl-5-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
6-cyclopentyl-1-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(1H-1,3-benzodiazol-1-yl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)propanamide
N,N-dimethyl-1-{[2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfonyl}pyrrolidin-3-amine
(4aS,8aR)-6-(5-propylthiophene-3-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
ethyl 2-{methyl[5-({[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amino}methyl)pyrimidin-2-yl]amino}acetate
(9aR)-8-(2-methoxybenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5,6-dimethyl-2-(2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
4-(hydroxymethyl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]azepan-4-ol
(1r,4r)-4-{[(2-methyl-1-benzofuran-5-yl)formamido]methyl}cyclohexane-1-carboxylic acid
3-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
2-(dimethyl-1,2-oxazol-4-yl)-2-[4-(2-methoxybenzoyl)piperazin-1-yl]acetic acid
N-cyclopropyl-2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
N-[(2,6-dimethylpyridin-4-yl)methyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
9-methoxy-7-(4-methoxyphenyl)-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclopentyl-N-[3-(2-fluorophenyl)propyl]-5-oxopyrrolidine-3-carboxamide
4-[(2,6-dichloro-3-hydroxyphenyl)methyl]-1,3-dimethylpiperazin-2-one
N-methyl-3-(5-methylthiophen-2-yl)-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
6-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2R,6R)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
2-{1-[(2-fluorophenyl)methyl]-4-(1,3-thiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[4-methyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenoxy]acetamide
N-tert-butyl-2-(pyridin-4-yl)benzene-1-sulfonamide
3-(2-amino-1,3-thiazol-4-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpropanamide
1-benzyl-5-{[(2,3-dimethoxyphenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-methyl-5-(5-phenyl-1,2-oxazol-3-yl)-1H-1,2,4-triazole
4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1-phenylpiperazin-2-one
2-ethyl-4-phenyl-9-(pyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one