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2-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}pyrrolidine-1-carboxamide
1-{4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-1,4-diazepan-1-yl}ethan-1-one
1-{1-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
N-(2-methylpropyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-(2-chlorophenyl)-N-(2-hydroxypropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
(1S,5S)-3-({4-methoxy-3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
5-(2-phenylethyl)-5-(piperidin-4-yl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
7-methyl-2-(5-methyl-4-phenylthiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]phenyl}-5-methyl-1H-1,2,3,4-tetrazole
1-{2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
2-[4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
5-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}-2,4,6-trimethylpyrimidine
4-(3-benzyl-1H-pyrazol-5-yl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine
1-[7-(furan-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-4-methyl-1,4-diazepane
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
4'-[2-(oxolan-3-yl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyrimidin-2-amine
(1R,6S)-N-[4-(3-acetylphenyl)phenyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
1-methyl-4-(3-methyl-3-phenylpiperidine-1-carbonyl)piperidin-4-ol
8-(3-fluoropyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(3-propoxypiperidin-1-yl)adamantan-1-ol
[(3R,4S)-1-[(3-chloro-2,6-difluorophenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-(dimethylamino)-2-(2-oxo-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-2,3-dihydropyridazin-3-one
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)pyridine-2-carboxamide
2-(4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}phenyl)pyridine
1-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
ethyl 1-[(2-chloro-6-methylphenyl)carbamoyl]-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
1-{2-[2-(butan-2-yl)phenoxy]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-methyl-5-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
8-acetyl-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1R,5R)-6-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
6-[3-(3-methylphenyl)piperidin-1-yl]pyridine-2-carboxylic acid
1,9-dimethyl-4-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(benzylsulfamoyl)[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]amine
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2,8-dimethyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]quinoline
3-[3-(piperidine-1-carbonyl)phenyl]-1-(1,2,3,4-tetrahydronaphthalen-1-yl)urea
4-({1-[(2-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperazin-2-one
2-{[3-(4-phenoxybenzoyl)piperidin-1-yl]methyl}pyridine
1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-6-ol
4-(4-fluorophenyl)-1-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}butan-1-one
1-(4-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}piperidin-1-yl)ethan-1-one
5-[(2E)-3-phenylprop-2-en-1-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(4-propanoylphenoxy)acetamide
(1R,5R)-6-[(2-fluoro-5-methoxyphenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-({2-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-(carbamoylmethyl)-N-[2-(pyridin-4-yl)ethyl]piperidine-4-carboxamide