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N,N,4-trimethyl-3-{[methyl(1H-pyrazol-3-ylmethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
6-cyano-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}pyridine-3-carboxamide
N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-[3-(oxolan-2-yl)propyl]acetamide
3-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-2,8-diazaspiro[4.5]decane
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-[5-(5-chlorofuran-2-yl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-ethyl-1-{[4-(2-methylphenyl)phenyl]methyl}-1,4-diazepan-5-one
N-benzyl-N-ethyl-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
(8R,9aS)-8-hydroxy-2-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
ethyl 4-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1-(pyrimidin-2-yl)piperidine-4-carboxamide
1-[1'-(5-ethylthiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-methyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}azepane-2-carboxamide
(4aS,8aR)-1-butyl-6-[3-(furan-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(3R,4R)-1-(cyclopent-1-ene-1-carbonyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
[(3R,4R)-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
propan-2-yl 2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
(1R,7S)-3-(2-ethylbutyl)-N-methyl-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(cyclohexylmethyl)-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
4-[(1H-1,3-benzodiazol-2-ylmethyl)sulfamoyl]-N-propylbenzamide
2-methyl-6-{2-[(thiolan-3-yl)amino]ethyl}-3,4-dihydropyrimidin-4-one
N-cyclopropyl-6-[4-(1H-pyrazol-1-yl)phenyl]pyridazin-3-amine
N-[1-(dimethylamino)propan-2-yl]-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
1-(2-methyl-5-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
4-methoxy-N-(4-{4-[({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]piperidin-1-yl}phenyl)benzamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylfuran-3-carboxamide
({4-ethyl-5-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(1-{4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-3-methylpiperidin-3-yl)methanol
1-(2-fluorophenyl)-4-[1-(thiophen-3-ylmethyl)piperidin-3-yl]piperazine
2-{[4-(4-methoxyphenyl)-5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
methyl 4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}benzoate
(2R)-2-amino-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-2-(thiophen-2-yl)acetamide
3-methyl-6-(oxolan-3-yl)-5-phenyl-1H-pyrazolo[3,4-b]pyridine
N'-(3-ethylphenyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)butanediamide
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-(cyclopentylmethyl)-N,6-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-dihydropyridine-3-carboxamide
1-cyclopropanecarbonyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N'1-[2-(dimethylamino)ethyl]-N'1-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopropane-1,1-dicarboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)formamido]ethyl}acetamide
4-(2-fluoro-5-methylphenoxy)-1-[2-(methylsulfanyl)propanoyl]piperidine-4-carboxylic acid
[(3-methoxyphenyl)methyl](prop-2-en-1-yl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
8-(1-benzoxepine-4-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
8-chloro-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
N-cyclopropyl-1-(methoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclobutane-1-carboxamide
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide