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2-(methylamino)-N-[1-(4-propylphenyl)ethyl]pyrimidine-5-carboxamide
8-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[2-(1H-1,2,4-triazol-1-yl)propyl]amine
N-cyclopropyl-6-[(1E)-pent-1-en-1-yl]pyridazin-3-amine
(1S,5R)-6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(1H-imidazol-1-yl)-1-(quinoline-2-carbonyl)piperidine-4-carboxylic acid
2-amino-1-[4-(4-{[cycloheptyl(ethyl)amino]methyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]ethan-1-one
2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-ethyl-4,6-dimethyl-3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1S,5R)-3-acetyl-N-[(2,4-dichlorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-methyl-7-(2-methyl-4-phenylpyridine-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
5-butyl-1-(3-phenylphenyl)-4-(pyridazine-3-carbonyl)piperazin-2-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(6-methyl-2-phenylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(3R,4R)-3-hydroxy-1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
(1R,2S)-N1-tert-butyl-N2-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}cyclohexane-1,2-dicarboxamide
1-ethyl-3-methyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]piperidine-3-carboxamide
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[(2-methylphenyl)methyl]urea
N3-methyl-N1-[4-methyl-3-(propan-2-yl)phenyl]pyrrolidine-1,3-dicarboxamide
(1R,5R)-6-[2-(2-methoxyphenoxy)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-[(pyridin-2-ylmethyl)amino]pyrrolidin-2-one
7-fluoro-2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
2-(2-{2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-6-chloro-2,3-dihydropyridazin-3-one
{[1-(2-fluorophenyl)cyclopropyl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
4-[(2-ethoxynaphthalen-1-yl)methyl]-2-(trifluoromethyl)morpholine
1-(4-benzylpiperazin-1-yl)-3-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-yl}propan-1-one
4-{4-[(3-methoxypyrrolidin-1-yl)methyl]phenyl}-2-methylbutan-2-ol
4-[3-(2-methoxyphenyl)propyl]-1,4-oxazepane
N-tert-butyl-2-(4-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenoxy)acetamide
1-(3-chlorophenyl)-4-[2-(3-hydroxyphenyl)acetyl]-5-methylpiperazin-2-one
4-phenoxy-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylic acid
4-(cyclopropylmethyl)-1-(4-methylpyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-(furan-2-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(2-methoxyphenyl)methyl]-11-(piperidin-1-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-ethyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
3-(ethoxymethyl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
2-(morpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(2-oxopiperidin-1-yl)acetamide
(1S)-S-[3-(azetidine-1-carbonyl)phenyl]-2-hydroxy-1-phenylethane-1-sulfonamido
({1-[(1-cycloheptanecarbonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)dimethylamine
methyl 5-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-[2-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenoxy]ethan-1-ol
4-{4-[(dimethylamino)methyl]phenyl}-2-methoxypyridine-3-carbonitrile
2-[5-(1-ethylpyrrolidin-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]quinoxaline
1-(3-methoxyphenyl)-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
1-[(2-fluorophenyl)methyl]-N-methyl-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4-{2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}butan-2-ol
N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide