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2-methoxy-3-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}pyridine
(2R,6R)-4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-methyl-5-{2-[(E)-2-phenylethenyl]phenyl}-1,3,4-oxadiazole
2-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3,4-dihydroquinazolin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-3-(morpholin-4-yl)propanamide
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-methyl-5-phenylpiperidin-2-one
5-[(isoquinolin-5-yloxy)methyl]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
3-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(2-fluorophenyl)-1H-indazol-1-yl]acetamide
2-{3-[4-(3-cyanophenyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-2-propyl-1,3-thiazole-4-carboxamide
9-hydroxy-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-cyclopropaneamido-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-methylbenzamide
1-[6-({1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}amino)pyridin-3-yl]ethan-1-one
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-3-methylfuran-2-carboxamide
N,3-dimethyl-4-oxo-N-(pyrimidin-4-ylmethyl)-3,4-dihydrophthalazine-1-carboxamide
(3aS,6aS)-2-acetyl-5-[4-(piperidin-1-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-methyl-4-(oxan-2-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
(3S,7S)-5-(2,6-diaminopyrimidin-4-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
N-{[3-(dimethylamino)phenyl]methyl}-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(morpholin-3-yl)acetamide
3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
8-fluoro-2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
N-(2-ethoxyethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N3-cyclooctyl-4-oxo-N5-[2-(propan-2-yloxy)ethyl]-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(2R,6S)-2,6-dimethyl-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]morpholine-4-carboxamide
4-{[(1S,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
(2R,6R)-4-{[6-(dimethylamino)pyridin-3-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-5-phenyl-1,2-oxazole-3-carboxamide
[1-(ethylsulfanyl)propan-2-yl]({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl})amine
2-methoxy-3-[3-(3-methoxyphenoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]pyridine
(1S)-1-{1-[2-(1H-imidazol-5-yl)ethyl]-3-methyl-1H-1,2,4-triazol-5-yl}-2-phenylethan-1-ol
3-(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-3-yl)-N-(2-fluorophenyl)propanamide
3-(4-methyl-1,3-thiazol-5-yl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
2-amino-N-[(2-chlorophenyl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-5-phenoxyfuran-2-carboxamide
1-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]urea
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[3-(1H-indol-1-yl)propyl]acetamide
1-(3-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
1-[(4-ethoxyphenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(2-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
(3aR,6aR)-2-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-cyclopropyl-1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-3-(thiophen-3-ylmethyl)urea