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N-{[4-(aminomethyl)phenyl]methyl}-3-(1-methyl-1H-pyrazol-5-yl)propanamide
3-methyl-6-{5-[1-(propan-2-yloxy)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
5-(2,3,4-trimethoxyphenyl)pyridine-3-carboxamide
1-(3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)propan-1-one
4-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[5-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-propoxyethan-1-one
5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
4-acetamido-N-{[4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]decan-4-one
3-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
2-[1'-(3-methylbut-2-en-1-yl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
(1R,3S)-3-(2-aminoethoxy)-7-(1-methyl-1H-indole-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-(propan-2-yloxy)-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridazine
3-[1-(2-fluorophenyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpropanamide
1-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
2-[1-(3-methylbutyl)-4-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
4-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]butanamide
3-butyl-1-{4-[4-(morpholine-4-carbonyl)pyridin-2-yl]phenyl}urea
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}propanamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-3-carbonitrile
5-(methoxymethyl)-3-({3-[3-(thiophen-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,2,4-oxadiazole
1-(2-{5-[(E)-2-(4-methoxyphenyl)ethenyl]-4-phenyl-1H-imidazol-1-yl}ethyl)piperidin-4-ol
3-(2-methoxyethyl)-1-(1H-1,2,3-triazol-4-ylmethyl)piperidine-3-carboxylic acid
6,7-dimethoxy-3-[(5-methylfuran-2-yl)methyl]-3,4-dihydroquinazolin-4-one
N-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(pyrimidin-4-yl)piperidine-1-carboxamide
3-(2-{3-hexyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[2-(adamantan-1-yl)-2-hydroxyethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[(2S)-2-(3,3-diphenylpiperidine-1-carbonyl)pyrrolidin-1-yl]ethan-1-one
(3R,4S)-4-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-amine
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
3-(3-fluorophenyl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1-hydroxy-2-methylpropan-2-yl)-1H-pyrazole-4-carboxamide
2-methoxy-4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(methylcarbamoyl)cyclohexyl]benzamide
5-(azepane-1-carbonyl)-N-cyclooctyl-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
4-methyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrimidine
N-[(3-chlorophenyl)methyl]-3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
1-[(1-{[1-(pyrazin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]azepane
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{4-[(2-ethyl-4-methyl-3-oxopiperazin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
N-benzyl-N-methyl-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-amine
3-(1H-imidazol-1-ylmethyl)-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
2-(dimethylamino)-N-[2-(1H-indol-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
4-[(4-fluorophenyl)methyl]-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidine
1-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-3-phenylpropan-1-ol
2-[2-(1H-pyrazol-1-yl)ethyl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
[2-(4-methoxyphenyl)ethyl][(4-methoxyphenyl)methyl][(1-methylpiperidin-4-yl)methyl]amine
methyl 2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetate