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N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-phenoxypropanamide
N-[(5-methylpyrazin-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
5-[1-(2-methoxyquinoline-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-(2,3-dimethylquinoxaline-6-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
1-cyclopentyl-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-methyl-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(dimethyl-1,3-thiazol-5-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
5-[4-(piperidin-3-ylmethyl)benzoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
(2S,4R)-4-hydroxy-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyrrolidine-2-carboxamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-3-amine
6-(2-fluoro-6-methoxyphenyl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
2-[3-(2,3-dihydro-1H-isoindol-2-yl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
(1R,5R)-3-methanesulfonyl-6-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1-benzofuran-5-carboxamide
(1S,5R)-3-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-4-(piperidin-1-ylmethyl)benzamide
9-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[3-cyclopropyl-5-(2-phenyl-1H-imidazol-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-(2-methoxyethyl)-1-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
8-(3-fluoropyridine-4-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(6-methoxypyrimidin-4-yl)piperazin-2-yl}ethan-1-ol
2,8-dimethyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}quinoline-4-carboxamide
N,N-dimethyl-2-{[(9H-purin-6-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[3-(3,4-diethoxyphenyl)propyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(2-phenoxyethyl)amino]methyl}phenoxy)propan-2-ol
(2S)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-cyclopropyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H-1,2,4-triazole
1-{2-[methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})amino]ethyl}piperidin-2-one
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
9-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
cyclopentyl 4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-amido}benzoate
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidin-3-ol
N-methyl-2-(methylamino)-N-[(4-phenoxyphenyl)methyl]-1,3-thiazole-4-carboxamide
1-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}naphthalen-2-ol
1-({1-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
5-[2-(difluoromethoxy)phenyl]-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
(3S,4S)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-ethyl-N,5-dimethyl-1,2-oxazole-4-carboxamide
1-[2-(2-chlorophenyl)ethyl]-N-[2-(1H-imidazol-1-yl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
9-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-({1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidin-3-yl}formamido)acetate
8-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)quinoline
1-(2-aminoethyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
2-(2-{[(1R,5R)-3-(dimethylcarbamoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)acetic acid
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-[4-(1-benzofuran-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]butanamide
2-methoxy-1-[1'-(pyridin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
ethyl 3-({5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazol-4-yl}formamido)propanoate