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5-(2-{4-[(4-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,3-dimethylimidazolidine-2,4-dione
N-cyclopropyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-amine
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-(3-methyloxetane-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
ethyl 1-{[5-(hydroxymethyl)furan-2-yl]methyl}-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]acetamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
3-(3-methyl-1H-pyrazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-benzyl-N,N-dimethyl-5-{[(4-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,6R)-3-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1,3-benzothiazole-6-carbonyl)pyrrolidin-3-yl]methanol
N-[2-(5-methylfuran-2-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N-(2-methoxyethyl)-5-methyl-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
(2R,4S)-4-hydroxy-1-[(6-phenoxypyridin-3-yl)methyl]piperidine-2-carboxylic acid
1-ethyl-N-(2-phenylethyl)-3-(propan-2-yl)-N-propyl-1H-pyrazole-5-carboxamide
2-(1-{[1-(quinoline-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-methoxybenzamide
N,4-dimethyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyrimidin-2-amine
N-(1-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
1-[(2S)-4,4-difluoropyrrolidine-2-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1-methylpiperidin-4-amine
N-[3-(4-fluorophenyl)phenyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-3-carboxamide
N-{2-[(1-methoxypropan-2-yl)amino]ethyl}-4-methylpyridin-2-amine
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]ethan-1-one
N-(4-chloro-3-methoxyphenyl)-2-{[(3S,4R)-4-ethoxyoxolan-3-yl]amino}acetamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(2-oxoazepan-3-yl)benzamide
methyl 1-{[7-(methylsulfanyl)-2-oxo-1,2-dihydroquinolin-3-yl]methyl}piperidine-4-carboxylate
2-[1-(cyclohexylmethyl)-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(3-chlorophenyl)-4-(isoquinoline-5-carbonyl)piperazin-2-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-[(4-methoxynaphthalen-1-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[1-(quinolin-2-ylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]piperidin-1-yl}ethan-1-one
(2E)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-3-yl)prop-2-en-1-one
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(1H-indol-3-yl)ethyl]acetamide
1-{[2-(carbamoylmethoxy)-5-chlorophenyl]methyl}-4-hydroxypiperidine-4-carboxylic acid
(4aS,7aR)-1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-hydroxyethyl)-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-hydroxyethyl)-N-[2-methyl-5-(3-methylbutanamido)phenyl]-3-oxopiperazine-1-carboxamide
6-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-methyl-N-[(1-methylpiperidin-3-yl)methyl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
2-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
2-(5-ethylthiophene-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2-(4-fluorophenyl)morpholine
(4aS,8aR)-1-(2-aminoethyl)-6-(4-methylquinolin-2-yl)-decahydro-1,6-naphthyridin-2-one
N-[(4-methoxyphenyl)methyl]-N,1-dipropyl-1H-pyrazole-5-carboxamide