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3-{[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenol
(furan-2-ylmethyl)(prop-2-en-1-yl){[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
N-(3-carbamoyl-4-methoxyphenyl)-4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carboxamide
1-(diphenylmethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2-{1-[4-(morpholin-4-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
ethyl(1H-imidazol-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}adamantan-1-ol
2-{4-[(3,4-dimethoxypyridin-2-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[4-(1H-pyrazol-3-yl)phenyl]sulfanyl}acetamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-hydroxyethan-1-one
2-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
4-(2-aminopyridine-4-carbonyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
2-(5-phenyl-1,3,4-thiadiazol-2-yl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-7-[(1R,2S)-2-propylcyclopropanecarbonyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2S)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
N-(oxolan-3-yl)-3-[(2,2,2-trifluoroethyl)sulfamoyl]benzamide
1-methyl-9-(prop-2-en-1-yl)-4-[2-(pyridin-3-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
N'-cyclopentyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)butanediamide
1,9-dimethyl-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)-1-(morpholin-4-yl)propan-1-one
(1S,4S)-2-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-2-azabicyclo[2.2.1]heptane
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
2-{[(3-methylthiophen-2-yl)methyl]amino}-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
2-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-N-methylacetamide
2-methyl-5-[4-({[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)piperidin-1-yl]-2,3-dihydropyridazin-3-one
N-[(2-fluorophenyl)methyl]-2-{[(2-phenyl-1,3-oxazol-4-yl)methyl]amino}acetamide
3-(2-fluorophenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-N-ethyl-1-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)pyrrolidine-2-carboxamide
1-(2-methoxyethyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrrolidine-3-carboxamide
8-methyl-2-[2-(pyridin-4-yl)pyrimidin-5-yl]-4-(pyrrolidine-1-carbonyl)quinoline
N-methyl-4-phenyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
2-amino-4-(2,3-dimethoxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-(thiophen-3-ylmethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
(4aS,8aR)-1-butyl-6-{[3-(pyridin-2-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
2-[(3-methoxyphenyl)amino]-N-(oxan-4-ylmethyl)butanamide
3-[(1S,2R)-2-aminocyclobutyl]-1-[(4-methylphenyl)methyl]urea
[(2-phenoxypyridin-3-yl)methyl](pyridin-2-ylmethyl)amine
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-methyl-5-phenylpiperidin-2-one
1-{2-methyl-5-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]phenyl}imidazolidin-2-one
({2-methoxy-5-[1-(pyridin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]phenyl}methyl)dimethylamine
N-methyl-3-phenoxy-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
(1S,5R)-N-(3-methylphenyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
8-(2-hydroxy-4-methoxybenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1,2-oxazole-5-carboxamide
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one