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2-(aminomethyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-1-carboxamide
N-methyl-2-(6-oxo-5,6-dihydrophenanthridin-5-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
7-(2-methoxyethyl)-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-{4-[4-(azocane-1-carbonyl)phenoxy]piperidin-1-yl}-3-methoxypropan-1-one
8-benzyl-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-acetyl-N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]benzamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-sulfonyl}-5-methyl-2,1,3-benzothiadiazole
N,N-diethyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
6-amino-2-(2-{[6-(piperidin-1-yl)pyrimidin-4-yl]amino}ethyl)pyrimidin-4-ol
2-chloro-N-[2-({2-oxo-1-oxaspiro[4.4]nonan-4-yl}formamido)ethyl]benzamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
1-(3-chlorophenyl)-4-(3-hydroxy-4-methylbenzoyl)piperazin-2-one
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
6-[2-(3,4-dichlorophenyl)morpholin-4-yl]pyrimidin-4-amine
2-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-2,3-dihydro-1,2-benzothiazol-3-one
4-(3-hydroxy-3-methylbutyl)-N-[2-(2-methyl-1H-indol-3-yl)ethyl]benzamide
5-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
methyl[(1-propyl-1H-imidazol-2-yl)methyl][2-(pyridin-2-yl)ethyl]amine
2-[2-(2-methoxyethoxy)acetyl]-N-methyl-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
5-[(benzyloxy)methyl]-1-[(3S,4R)-4-methoxyoxolan-3-yl]-4-phenyl-1H-imidazole
1-[(2-{[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]methyl}phenyl)methyl]pyrrolidin-2-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pent-4-enamide
(4aS,7aR)-1-(1-methyl-1H-pyrazole-3-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-cyclopropyl-2-(1H-imidazol-2-yl)-N-[(3-methoxyphenyl)methyl]benzamide
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})(2-phenylethyl)amine
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
3-methyl-N-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
ethyl 4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine-1-carboxylate
1-(2-methylpentyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
7-(2,6-dimethoxypyrimidine-4-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(2-methoxyphenyl)methyl]-2-(1-methylpiperidin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
6-[6-hydroxy-4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyrazine-2-carboxamide
8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(2S)-2-(2-{5-[(4-chlorophenyl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)propanamide
4,4,4-trifluoro-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}butanamide
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-methyl-1,2-dihydroquinoxalin-2-one
[(4aS,8aR)-6-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-4a-yl]methanol
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(1-hydroxy-3-methylbutan-2-yl)-1,3-oxazole-4-carboxamide
6-methyl-1-(prop-2-en-1-yl)-3-{[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-fluorophenyl)methyl]piperidine
2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
4-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
4-benzyl-1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1,4-diazepan-5-one
1-methyl-4-[({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]piperidin-4-ol
methyl (2S,4S)-1-benzyl-4-(5-chloro-3-phenyl-1H-indole-2-amido)pyrrolidine-2-carboxylate
2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}benzoic acid
5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-2-fluorobenzamide
1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-(methoxymethyl)piperidine