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N-{2-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-2-yl]ethyl}acetamide
N-(2-methoxyethyl)-2-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)propanamide
1-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydroquinoline
methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})[(2,4,5-trimethylphenyl)methyl]amine
(3S,4R)-1-(4-methoxy-3-methylbenzoyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
(3R,4R)-1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-cyclobutyl-4-methylpyrrolidin-3-ol
2-({4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanamide
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-(azepan-1-yl)-1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)butan-1-one
6-chloro-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methyl-1H-indole-2-carboxamide
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-methyl-4-oxo-2-(phenoxymethyl)-N-phenyl-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
2-[5-(2,3-difluorophenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-[4-({methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenyl]ethan-1-amine
3-chloro-4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
3-{[4-(4-methoxybenzenesulfonyl)piperazin-1-yl]methyl}pyrrolidin-3-ol
4-[(dimethylamino)methyl]-1-(quinoxalin-2-yl)azepan-4-ol
N-(2-hydroxyethyl)-3-{imidazo[1,2-a]pyridin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanamide
1-(1-propylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
(3S,4S)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
1-{[1-(4-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
dimethyl[(4-methyl-5-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-methyl-1,4-diazepan-5-one
4-(5-hydroxypyrazine-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 3-benzyl-1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperidine-3-carboxylate
N-[4-(2-fluorophenoxy)phenyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxamide
3-(2,3-dihydro-1H-isoindol-2-yl)-1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}propan-1-one
4-cyclobutyl-N,6-dimethyl-N-[2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
2-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-imidazole
(4aS,8aR)-1-(2-phenylethyl)-6-(2-propoxyacetyl)-decahydro-1,6-naphthyridin-2-one
4-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyrimidine-5-carboxylic acid
1-tert-butyl-5-oxo-N-[3-(pyridin-2-yl)propyl]pyrrolidine-3-carboxamide
2-(1-propyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-3-methoxypyrazine
1-[cyclohexyl(methyl)amino]-3-[4-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol
1-{2-[(3R,4S)-3-[(2-methylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
3-(pyridin-4-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-{[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzoic acid
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-[methyl(propan-2-yl)amino]ethan-1-one
3-(4-hydroxyphenyl)-N-[2-(propane-2-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
4-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-1-phenylpiperazin-2-one
8-methyl-2-propyl-3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
N-[(1R,3S)-3-(morpholine-4-carbonyl)cyclopentyl]-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
(1R,3S)-3-{[(3-chloro-2-methylphenyl)methyl]carbamoyl}cyclopentane-1-carboxylic acid
methyl 4-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pentanoate
1-(furan-2-ylmethyl)-N-[(6-methylquinolin-5-yl)methyl]piperidine-4-carboxamide
3-(5-methyl-1H-pyrazol-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpropanamide
2-[7-(hydroxymethyl)-9-(pyrimidin-2-yl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-ol