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[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](2-methylpropyl)(pyridin-2-ylmethyl)amine
2-{[(3-ethoxyphenyl)methyl]({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})amino}ethan-1-ol
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-amino-6-(5-chlorothiophen-2-yl)-5-methyl-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-4-carboxamide
4-[3-(4-benzylpiperazine-1-carbonyl)phenyl]-2-methylbutan-2-ol
3-chloro-4-hydroxy-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}benzamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)morpholine-2-carboxamide
(1R,7S)-3-(4-fluoro-2-methylphenyl)-N-methyl-4-oxo-N-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-methyl-4-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
[(2S,6S)-4-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
methyl 2-hydroxy-5-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]benzoate
N-[1-(methoxymethyl)cyclopentyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}(2-phenylethyl)amine
6-methyl-3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(4-methylphenyl)ethyl]benzamide
(4aR,7aS)-1-ethyl-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)acetamide
3-(3-methoxypropyl)-1-(1H-1,2,4-triazole-5-carbonyl)piperidine-3-carboxylic acid
(1S,5R)-3-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclopentyl-3-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
dimethyl[(4-methyl-5-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(2,6-dimethylpyridin-3-yl)pyrimidine
2-({[3-(dimethylamino)thiolan-3-yl]methyl}amino)-N-[2-(4-fluorophenyl)ethyl]acetamide
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-methyl-1-(2-methyl-5-sulfamoylphenyl)urea
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[4-(trifluoromethyl)phenyl]methyl}amine
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(1H-pyrazol-1-yl)butanamide
9-[(4-fluoro-3-methylphenyl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N,1-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
1-methyl-5-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]piperidin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-methyl-N-(oxan-2-ylmethyl)-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-ethyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,4-dihydroquinolin-4-one
2,3-dimethyl-N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}-1H-indole-5-carboxamide
1-[2-(dimethylamino)-4-{[(5-fluoro-1H-indol-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-(azocan-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-[4-(4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-1-yl)phenyl]ethan-1-one
(5S,9aS,9bS)-5-[(E)-2-(furan-2-yl)ethenyl]-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
2-({4-[4-(4-methoxypiperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-{4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1H-pyrrole-2-carbonyl)piperidine
2-({4-[5-(piperidine-1-carbonyl)furan-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
5-methoxy-N-[2-(4-methylmorpholin-2-yl)ethyl]-1H-indole-2-carboxamide
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-[2-(5-methylfuran-2-yl)propyl]-1H-1,2,3-triazole