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5-chloro-3-methyl-2-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1H-indole
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(pyridin-4-yl)propan-1-one
3-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(pyridine-3-carbonyl)pyrrolidine-2-carboxamide
1-ethyl-N-pentyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pentan-1-one
3-(cyclobutylmethoxy)-5-[(pyridin-4-ylmethyl)carbamoyl]benzoic acid
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(1H-imidazol-1-ylmethyl)piperidine-1-carboxamide
2-[5-(azocan-1-ylmethyl)-3-cyclopentyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]-1-[(4-methylphenyl)methyl]piperazin-2-one
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
N-[1-(hydroxymethyl)cyclopentyl]-3-(4-hydroxyphenyl)benzamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
1,4,6-trimethyl-2-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
1-methyl-4-{1-[(3,4,5-trimethoxyphenyl)methyl]-1H-imidazol-2-yl}piperidine
N-benzyl-N-methyl-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
2-amino-6-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-4-(piperidin-4-yl)pyridine-3-carbonitrile
(2S,4R)-1-(cyclohexylmethyl)-N-(propan-2-yl)-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
2-{2-[(3S)-3-ethylmorpholin-4-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
N,N-dimethyl-3-[3-(2-methyl-1,3-thiazol-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]propanamide
4-({methyl[2-(2-methylpiperidin-1-yl)ethyl]amino}methyl)benzoic acid
1-{2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
1-{2-[1-benzyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine
5-{[2-(4-chlorophenyl)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(3-ethylphenoxy)ethyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)propanamide
3-(2-oxo-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-[(3-fluoropyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
8-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(2E)-3-(furan-2-yl)prop-2-en-1-yl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
7-[cyclohexyl(methoxy)methyl]-4-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{5-[5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]furan-2-yl}benzonitrile
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(2-methylphenyl)-1H-pyrazole
(3S)-1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-fluoropyrrolidine
N-(3-hydroxypropyl)-3-(1H-imidazol-2-yl)-N-(pyridin-4-ylmethyl)benzamide
4-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-1,4-oxazepan-6-ol
3-methyl-7-[2-(2-methylphenyl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
ethyl 5-(1H-indole-3-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[3-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(1H-imidazol-1-yl)-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
2-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)amino}methyl)phenol
14-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
methyl[(3-methylthiophen-2-yl)methyl]{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine
2-(2,4-dimethoxyphenyl)-4-[1-(pyridine-3-carbonyl)pyrrolidin-3-yl]pyridine
4-(1H-pyrazol-4-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]butan-1-one
ethyl 1-(1-ethylpiperidin-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
methyl 3-{[5-benzyl-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate