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(morpholin-2-ylmethyl)({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
(2R)-2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}pentanediamide
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-(5-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-[2-(2-chlorophenoxy)ethyl]-2-hydroxybutanamide
2-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}benzamide
2-ethyl-9-[(6-methylpyridin-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-({[(propan-2-yl)carbamoyl]methyl}carbamoyl)pyrrolidine-2-carboxylic acid
N-cyclopropyl-4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazine-2-carboxamide
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-ol
N-(2-hydroxyethyl)-2,2-dimethyl-N-[(5-methylthiophen-2-yl)methyl]oxane-4-carboxamide
2-(morpholin-3-yl)-1-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}ethan-1-one
(1s,4s)-4-{4-[2-(1-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
3-[3-({[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
1-{4-[2-(pyridin-3-yl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
(3S,4S)-1-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}piperidine-3,4-diol
N-(1-benzylpyrrolidin-3-yl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2-aminoacetyl)-N-(cyclopropylmethyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
5-[3-(1H-imidazol-1-yl)propyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4,4-difluoro-N-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]piperidine-1-carboxamide
2-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamide
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(dicyclopropylmethyl)methylamine
6-(2-chlorophenyl)-7-methyl-2-(piperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-methoxy-N-{3-[1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}acetamide
2-{2-[5-(4,5-dimethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrazine
5-[4-(2-hydroxypropan-2-yl)piperidin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-2-hydroxybenzoic acid
3-(2,1,3-benzothiadiazol-5-ylmethyl)-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-(2-hydroxyacetyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
4-methyl-9-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
5-hydroxy-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}pyrazine-2-carboxamide
(4aS,8aR)-6-[(2-fluoro-4-methoxyphenyl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
ethyl 1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-methoxyethyl)piperidine-4-carboxylate
N-(3-{2,7-diazaspiro[4.5]decane-2-carbonyl}-2-methylphenyl)furan-2-carboxamide
2-methyl-N-{1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-{[7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1-benzofuran-2-carboxamide
2-(1H-pyrazol-1-yl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]butan-1-one
2-(dimethylamino)-N-(1-ethylcyclopropyl)-2-(3-methylphenyl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-2-(3-ethyl-1H-pyrazol-5-yl)-1H-imidazole
6-[(diethylamino)methyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{4-[2-(4-chlorophenoxy)ethyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetic acid
3-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]pyridin-2-ol
4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)-N-(1-propyl-1H-1,2,3-triazol-4-yl)piperazine-1-carboxamide
(2S)-2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-hydroxypropanamide
(3S,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[3-(cyclohexyloxy)propyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide