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N-butyl-2-[1-(2,6-dimethylpyridin-4-yl)-N-methylformamido]acetamide
3-methyl-1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroquinazolin-2-one
5-chloro-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
N-tert-butyl-2-{2-[2-(dimethylamino)ethoxy]phenyl}benzene-1-sulfonamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-(furan-2-ylmethyl)-5-{1-[2-(1H-pyrazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-benzyl-1-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]piperidine-3-carboxamide
2-[4-(2-aminopyridine-4-carbonyl)piperazin-1-yl]-N-ethylacetamide
2-{[5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)pyridin-2-yl](methyl)amino}ethan-1-ol
7-[2-(1H-pyrazol-1-yl)butanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5,7-dimethyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-{1-butyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}propanamide
4-[(2-methylphenyl)sulfanyl]-1-(1H-pyrrole-2-carbonyl)piperidine
1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-3-(2-methoxybenzoyl)piperidine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1-(oxan-4-yl)piperidine-3-carboxamide
1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
8-[3-(4-hydroxyphenyl)propanoyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3-oxazolidin-2-one
3-{5-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-{5-chloro-2-[4-(2-propoxyethyl)piperazine-1-carbonyl]phenyl}propanamide
1-methyl-5-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
4-(5-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}pyridin-2-yl)morpholine
N-ethyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-(pyridin-4-ylmethyl)acetamide
6-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(pyridin-3-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-{[5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)pyridin-2-yl]amino}propan-1-ol
4-[3-(difluoromethoxy)benzoyl]-1-(1H-indazol-6-yl)-5-methylpiperazin-2-one
1,3,6-trimethyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{2-[1-(1,3-thiazol-4-ylmethyl)piperidin-2-yl]ethyl}phenol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-[(3R,4S)-1-[(1-methyl-1H-indol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinolin-4-ylmethyl)amine
N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]-2,3-dihydro-1-benzofuran-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-phenylpiperazine
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
2-(2-methylpropyl)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-{[1-(3-chloro-4-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-methyl-N-(1,2-oxazol-5-ylmethyl)-3-(piperidin-4-ylmethyl)benzamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzamide
2-{[6-(8-methylquinolin-5-yl)pyrazin-2-yl]sulfanyl}acetic acid
N-(2,3-dihydro-1H-inden-2-yl)-6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(2,5-dimethylfuran-3-carbonyl)-4-(pyridin-3-ylmethyl)piperazine
1-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
N-[(3R,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
(4S)-1-(1H-imidazol-4-ylmethyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
5-{[(4-hydroxyphenyl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-cyclopentyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-oxopyrrolidine-3-carboxamide