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ethyl (4aS,8aR)-6-[(4-fluorophenyl)methanesulfonyl]-decahydro-1,6-naphthyridine-4a-carboxylate
(1S,5R)-6-(2-methoxyethyl)-3-{[3-(trifluoromethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(oxolan-2-ylmethyl)-3-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
7-chloro-1-methyl-2-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1H-indole
4-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(3S,4R)-N,N-dimethyl-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-4-(4-methylphenyl)pyrrolidin-3-amine
7-fluoro-2-methyl-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}quinoline-4-carboxamide
N-({1-[(4-tert-butylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-hydroxyacetamide
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]pyridine-2-carboxamide
3-phenyl-N-[1-(2-phenylethyl)piperidin-3-yl]prop-2-ynamide
3-[(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzonitrile
N-[1-(1-methylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-(3-phenyl-1H-pyrazol-1-yl)acetamide
2-(4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
ethyl 1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
3-(1-ethyl-1H-pyrazol-4-yl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
4-{2-[({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]ethyl}phenol
4-(4-chlorophenoxy)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidine
N-({1-[(dimethyl-1,3-thiazol-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-2-methoxyacetamide
3-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methoxybenzoic acid
2-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
(2R,6R)-4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[(3R,4S)-1-(4-fluoro-3-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1,3-dimethyl-2,6-dioxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N4-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(3-{thieno[2,3-d]pyrimidin-4-yl}phenyl)methanol
5-(1H-imidazol-2-yl)-1-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-phenyl-1H-imidazole
3-{[(butan-2-yl)amino]methyl}-2-methoxy-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)cyclohexanecarboxamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-(1H-pyrazol-1-yl)benzamide
(3aS,6aS)-1-[5-(benzyloxy)-2-methyl-1-benzofuran-3-carbonyl]-octahydropyrrolo[2,3-c]pyrrole
5-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]-1H-1,2,3-benzotriazole
1'-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[4-(2-fluorophenyl)phenyl]methyl}pyrrolidin-3-yl]methanol
4-[6-(methoxymethyl)pyrimidin-4-yl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(dimethylamino)azepan-1-yl]-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-benzoyl-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazine
(3S,4R)-1-[1-(methoxymethyl)cyclopropanecarbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(1R,2R)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-phenylcyclopropane-1-carboxamide
1-[(3-fluorophenyl)methyl]-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
ethyl 2-[4-({[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]carbamoyl}amino)phenyl]acetate
2-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]quinoline
4-(2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)morpholine-3,5-dione
N,1-dimethyl-3-(2-methylpropyl)-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
2-(5-acetylthiophen-3-yl)-1-[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]ethan-1-one
2-(2-phenylethyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidine
6-methoxy-2-oxo-N-[4-(pyridin-2-yl)butyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
[(2S,4R)-1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)-4-(dimethylamino)pyrrolidin-2-yl]methanol
3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea