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2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanamide
N-{1-[(5-propylfuran-2-yl)methyl]piperidin-3-yl}acetamide
(3R,4R)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
4-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
(3aR,6aR)-2-methanesulfonyl-5-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-{[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenyl)ethan-1-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclopentanecarboxamide
1-[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
4-hydroxy-N-[3-(phenylsulfanyl)propyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
2-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(dimethyl-1,2-oxazol-4-yl)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)pyrrolidine-1-carboxamide
4-benzyl-3-ethyl-1-(pyridazine-3-carbonyl)-1,4-diazepan-5-one
9-(2-methoxyethyl)-1-methyl-4-(1,2-oxazole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methoxy-1-[4-(4-methylphenoxy)piperidin-1-yl]ethan-1-one
2-(adamantan-1-yl)-N-methyl-N-[4-(morpholin-4-yl)butyl]acetamide
2-{[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
4-chloro-2-[3-(1H-pyrazol-3-yl)phenyl]aniline
N-butyl-3-{3H-imidazo[4,5-b]pyridin-6-yl}benzamide
2-ethoxy-6-({3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
N-[2-(2-methoxyphenyl)ethyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)phenol
methyl 4-({4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)benzoate
(5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-indol-2-yl)methanol
9-methoxy-4-[(2-methoxyphenyl)methyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-(4-methoxyphenyl)ethan-1-one
N-(furan-2-ylmethyl)-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-(adamantan-1-yl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylacetamide
methyl 6-(3,3-dimethylbutanoyl)-2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[4-(1H-imidazol-1-yl)phenyl]-1-[2-(propan-2-ylsulfanyl)ethyl]-1H-imidazole
(1,3-benzoxazol-2-ylmethyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-4-(furan-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
1-methyl-3-(propan-2-yl)-N-[4-(pyridin-2-yl)butyl]-1H-pyrazole-5-carboxamide
[(3S,4S)-4-(hydroxymethyl)-1-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl]methanol
N-(2,3-dihydro-1H-inden-1-yl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-methyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}cyclohexanecarboxamide
4-{4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-{4-[(4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}-N-(pyridin-3-yl)acetamide
3-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-2-yl}pyridine
1-({1-[1-(6-chloropyridin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)-1,4-diazepane
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]pyridine-3-carboxamide
5-[(6-ethoxyquinolin-2-yl)methyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[4-(furan-2-yl)butan-2-yl]urea
1-(2-{2-tert-butyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}ethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-methoxy-1-{1'-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-[4-(4-tert-butylphenyl)butanoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
5-(4-chloro-1-methyl-1H-pyrrol-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole