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N-[2-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)quinolin-6-yl]acetamide
N-benzyl[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)amino]sulfonamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]acetamide
1,3,6-trimethyl-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-chloro-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
(3aS,6aS)-2-propyl-5-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-1-(2-methylpropyl)-1H-1,3-benzodiazole
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(4-methylmorpholin-2-yl)ethyl]propanamide
1-(2-fluorophenyl)-4-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
(4aS,8aR)-6-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[3-(benzyloxy)phenyl]-3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]urea
1-(2-oxo-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-(propan-2-yl)piperidine-3-carboxamide
2-(2-{[1-(cyclopropylmethyl)-7-oxoazepan-4-yl]amino}ethyl)-1,2,3,4-tetrahydrophthalazine-1,4-dione
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
N-phenyl-3-(4-phenylbenzoyl)piperidine-1-carboxamide
(1S,5R)-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({4-hydroxy-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]azepan-4-yl}methyl)methanesulfonamide
2-[(4-chlorophenyl)methyl]-8-(thiophen-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
1-{6-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
N-ethyl-N-(2-hydroxyethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S,4R)-4-amino-1-{[4-(3,4-dimethylphenoxy)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
2-(1-methylpiperidin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
5-(2-methyl-3-phenylcycloprop-2-ene-1-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylpropanamide
1-(2-methoxyphenyl)-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazole
N-[3-(1H-imidazol-1-yl)propyl]-2-methanesulfonyl-N-(pyridin-3-ylmethyl)acetamide
2-(2-oxo-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)benzonitrile
2-(4-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}piperazin-1-yl)-N-ethylacetamide
4-chloro-N,1-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
3-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
2-[methyl(1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}piperidin-4-yl)amino]ethan-1-ol
1-(3-phenylpropyl)-5-(thiomorpholine-4-carbonyl)piperidin-2-one
4-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-(2-{4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}ethyl)phenol
3-(3-hydroxy-3-methylbutyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
6-methoxy-3-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1-benzofuran-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-[1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]methanesulfonamide
3-(4-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)prop-2-yn-1-ol
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[(2-fluorophenyl)methyl]-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-5-one
(4aR,6R,8aS)-2-(5-chloro-3-fluoropyridin-2-yl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-[2-(5-methylfuran-2-yl)ethyl]-3-(piperidin-3-yl)benzamide
1-[5-({[2-(1-hydroxycyclopentyl)ethyl](methyl)amino}methyl)-1-methyl-1H-pyrrol-3-yl]ethan-1-one
3-cyclopropyl-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide