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1-(4-methoxyphenyl)-3-(2-methylpropyl)-5-(oxan-4-yl)-1H-1,2,4-triazole
methyl 3-{1-[2-(2-oxoazonan-1-yl)acetyl]piperidin-4-yl}propanoate
methyl 3-{[4-(2-acetylbenzoyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-ethyl-1H-pyrazole-3-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(thiophen-2-ylformamido)pentanamide
1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(propan-2-yl)-1H-imidazole
6-({cyclohexyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methylurea
N-[(1S,2R)-2-carbamoylcyclopentyl]-3-(3-hydroxy-3-methylbutyl)benzamide
7-(5-methylthiophen-2-yl)-4-[(2R)-oxolane-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1'-{imidazo[1,2-a]pyridine-3-carbonyl}-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
5-(methoxymethyl)-N-(1-phenylbutyl)furan-2-carboxamide
(4aR,7aS)-1-ethyl-4-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(morpholin-4-yl)benzamide
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[1-(4-methylpyridin-2-yl)propyl]acetamide
N-(2H-1,3-benzodioxol-5-yl)-1-[(1,2-dimethyl-1H-indol-3-yl)methyl]piperidin-3-amine
6-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2,2-dimethyl-N-(2-methylpropyl)oxane-4-carboxamide
5-{3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
7-chloro-4-(3,5-difluoropyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(4-chlorophenyl)methyl]-4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carboxamide
4-chloro-1-methyl-3-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]-1H-indazole
N-(1,3-dihydroxy-2-methylpropan-2-yl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-fluoro-N-{1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-(4-{[1-(2-methoxyethyl)-2,4-dioxo-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
methyl 3-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]propanoate
(3R,4S)-4-(3-methoxyphenyl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-amine
2-cyano-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(4-methoxyphenyl)furan-2-carboxamide
N-[2-(dimethylamino)ethyl]-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]propanamide
(2S,4R)-1-benzyl-4-(cycloheptylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2S,4R)-N-ethyl-1-[(3-hydroxyphenyl)methyl]-4-(oxane-4-amido)pyrrolidine-2-carboxamide
4-(azepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)quinoline
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4-phenoxybutan-1-one
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-(2,3-dihydro-1H-inden-2-yl)piperazin-2-one
4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
[(3R,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(3-methylpyridin-4-yl)-4-{pyrazolo[1,5-a]pyridine-7-carbonyl}-1,4-diazepane
(3S,4S)-4-cyclopropyl-1-[(3-fluoro-4-methoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
3-[1-(2-hydroxyethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
3-[2-(2-hydroxyethoxy)ethyl]-1-(5-methoxy-2-methylphenyl)urea
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1H-pyrazole-4-carboxamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
5-{[4-(3-ethylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}isoquinoline
1-(2-ethoxyethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)benzoic acid
3-ethyl-N-[2-(4-methoxyphenyl)ethyl]-N-(oxolan-2-ylmethyl)-1,2-oxazole-5-carboxamide