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1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}azetidin-3-ol
2-({[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]amino}methyl)-6,8-dimethylquinolin-4-ol
7-cyclohexyl-2-(3-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
5-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(oxan-4-yl)piperidin-4-yl]-3-propyl-1H-pyrazole-5-carboxamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1R,3R)-3-aminocyclopentyl]-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
2-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidin-1-yl]acetic acid
N-ethyl-3-(1-methyl-1H-pyrrol-2-yl)-N-[2-(phenylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
1-{2-[methyl({[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino]ethyl}piperidin-2-one
[(3R,4R)-1-(3,5-difluorobenzoyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
ethyl 1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-{[2-(carbamoylmethyl)piperidin-1-yl]sulfonyl}-N-cyclobutylbenzamide
4-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]piperazin-2-one
1-(4-fluoro-2-methylphenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-amine
methyl 3-({1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidin-4-yl}formamido)propanoate
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
3-[3-(propan-2-yloxy)phenyl]pyridin-2-ol
7-[(2-fluorophenyl)methyl]-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[3-(2-fluorophenyl)pyrrolidin-1-yl]-6-methoxypyrimidin-2-amine
2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propane-1,3-diol
3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
5-fluoro-2-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-{1'-benzoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
1-[1-(3-chlorobenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-ethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(1S)-1-phenylethyl]-1,2-oxazole-3-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
2-methyl-7-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-amino-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}cyclopropane-1-carboxamide
1-(3-fluorophenyl)-6,6-dimethyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-{[4-(2,5-dimethylphenyl)-1H-1,2,3-triazol-1-yl]methyl}-2,1,3-benzoxadiazole
6-(2-hydroxyethyl)-N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
2-cyclopropyl-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]pyrimidine-5-carboxamide
2-(3-acetyl-1H-indol-1-yl)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylbutanamide
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
ethyl 3-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)propanoate
8-[(2-chloro-6-methylphenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[2-(2-chloro-4-methylphenoxy)ethyl]benzene-1-sulfonamide
7-methoxy-3-(pyrimidin-2-ylmethyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
5-[({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-N,N-dimethylpyrimidin-2-amine
2-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
(3S,9aR)-3-(cyclohexylmethyl)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione