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2-methoxy-4-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
N-[2-(furan-2-yl)ethyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}benzoic acid
2-chloro-4-{[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}-6-methoxyphenol
1-{1-[3-(methoxymethyl)piperidin-1-yl]propan-2-yl}-1H-1,3-benzodiazole
(2S,4R)-N,N-diethyl-1-(furan-3-ylmethyl)-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
methyl (2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
9-[2-(propan-2-yloxy)propanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-1-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]piperidine-4-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,4-dimethyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
6-(cyclopropylmethoxy)-1-(pyridin-3-ylmethyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
3-{[(3,4-dimethoxypyridin-2-yl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
2-(2-hydroxyphenoxy)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
2-[1-(2-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N4-benzyl-7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-benzyl-2-(3-methyl-2-oxopyrrolidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
4-chloro-N-(2-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}ethyl)benzene-1-sulfonamide
1-(3-methoxyphenyl)-2,2-dimethyl-4-(1H-pyrazole-4-carbonyl)piperazine
dimethyl({2-[2-(1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]ethyl})amine
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(3-ethyl-1,2-oxazol-5-yl)methyl]amine
3-[3-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propyl]pyridine
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(4-fluorophenoxymethyl)-4-hydroxypyrimidine-5-carboxamide
4-(3,5-dichloro-4-methylbenzoyl)-2-(2-methoxyethyl)morpholine
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(4-fluorophenyl)morpholine
2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-methylpyrimidin-4-amine
3-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
3-[4-(4-methylpiperazin-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]propanamide
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-1-methyl-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}morpholine-2-carboxamide
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
7-[(1-methyl-1H-indol-5-yl)methyl]-2,7-diazaspiro[4.5]decane
1-(2-methoxyethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylpyrrolidine-3-carboxamide
1-methyl-4-phenyl-3-({1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(thiophen-2-yl)ethan-1-one
methyl (2S,4S)-4-[2-hydroxy-6-(trifluoromethyl)pyridine-3-amido]-1-methylpyrrolidine-2-carboxylate
3-(2-fluorophenyl)-3-phenyl-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
[1-(4-chlorophenyl)propan-2-yl]({1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N,8-dimethyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[(2-methylphenyl)sulfanyl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
5-methyl-1-(4-{4-[(oxan-4-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
2-(phenoxymethyl)-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-ethyl-3,6-dimethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1-benzofuran-2-carboxamide
2-[({1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}oxy)methyl]pyridine
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidin-3-yl]cyclopropanecarboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methylacetamide
N-[3-(dimethylamino)propyl]-5-(methoxymethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(1R,3S)-3-(4-{[3-(trifluoromethyl)phenyl]methyl}piperazine-1-carbonyl)cyclopentan-1-amine