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N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
2-(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
2-{5-[3-(carbamoylmethoxy)phenyl]-4-phenyl-1H-imidazol-1-yl}acetic acid
1-methyl-3-(pyridin-3-ylmethyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-propyl-1,3,4-oxadiazol-2-amine
N-({1-[(E)-2-phenylethenesulfonyl]piperidin-3-yl}methyl)furan-2-carboxamide
[(2S,6S)-4-[5-(ethylsulfanyl)thiophene-2-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-[3-({[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
4-(2,5-dimethylbenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
2-methyl-8-{2-[(4-methylphenyl)methyl]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
(2R,6S)-2,6-dimethyl-4-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)morpholine
(3S,4S)-4-(propan-2-yl)-1-(propylcarbamoyl)pyrrolidine-3-carboxylic acid
4-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-methyl-1H-imidazole
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-ethyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[3-(hydroxymethyl)piperidin-1-yl]methyl}-N-(isoquinolin-1-yl)benzamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methylacetamide
N-cyclopropyl-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-(4-methylphenoxy)piperidine
1-(2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
(1S,4S)-5-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl 2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidine-1-carbonyl]amino}benzoate
N-cyclobutyl-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)thiophene-2-carboxamide
9-(2-hydroxypyridine-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(but-3-enoyl)-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(6-{1,4-diazabicyclo[3.2.2]nonan-4-yl}-2-methylpyrimidin-4-yl)ethan-1-amine
7-(3-cyclopropylpropanoyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N'-(2-methylphenyl)-N-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}propanediamide
4-ethyl-3-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}pyrrolidin-2-one
1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(1H-pyrazol-1-yl)propan-1-one
2-methyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
3-(1,4-diazepane-1-sulfonyl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)propanamide
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}benzamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-{[2-methyl-2-(morpholin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]urea
2-methoxyethyl 9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-{1-[(3-methoxyphenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2-(dimethyl-1,3-thiazol-5-yl)-N-[1-(thian-4-yl)piperidin-4-yl]acetamide
N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(2,5-dimethylbenzenesulfonamido)acetic acid
3-{1-[(2-phenylphenyl)methyl]azetidin-3-yl}pyridine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-methyl-6-oxo-N-[1-(phenylcarbamoyl)piperidin-4-yl]-1,6-dihydropyridine-3-carboxamide
2-{2-chloro-4-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}acetamide