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N,4-dimethyl-2-(methylamino)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-{4-[2-(morpholin-4-yl)ethyl]piperazin-1-yl}ethan-1-one
9-(5-phenyl-1,2,4-oxadiazol-3-yl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine
4-({4-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
(3aS,6aS)-5-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}pyrimidine
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-hydroxyacetamide
4-[(1-methyl-1H-imidazol-2-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-N,N-dimethylpropanamide
4-({5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
(2S,4S)-4-amino-1-(butane-1-sulfonyl)-N-methylpyrrolidine-2-carboxamide
4-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1H-indole
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
8-(3-carboxy-6-methylpyridin-2-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1,8-naphthyridine
{2-[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]-1,3-thiazol-4-yl}methanol
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
9-(3-fluoro-4-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3-(cyclopentyloxy)phenyl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-{1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-yl}acetamide
(1s,4s)-N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxycyclohexane-1-carboxamide
2-cyclopropyl-9-(4-methylpyrimidin-2-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-tert-butyl-N-[3-(4-chlorophenoxy)propyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
2-[5-(ethanesulfonyl)thiophen-2-yl]-1-benzofuran
2-[1-({3-ethoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)azetidin-3-yl]pyridine
N-(2-methoxyethyl)-1-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(piperidin-1-ylmethyl)piperidine
7-fluoro-2-methyl-4-[2-(trifluoromethyl)morpholine-4-carbonyl]quinoline
1-cyclohexyl-4-(oxolane-2-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N'-(2,5-dimethylphenyl)-N-(1-propylcyclopropyl)propanediamide
(2S,4R)-4-({[3-(benzyloxy)phenyl]methyl}amino)-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
3-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
4-(2,6-dimethylpyridin-3-yl)-N-[2-(oxolan-3-yl)ethyl]pyrimidin-2-amine
2-(4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazin-1-yl)-1,3-benzothiazole
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
2-({2-amino-6-[4-(1H-pyrazol-5-yl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-methyl-1,3-thiazole
5-[(4-fluoro-3-methylphenyl)methyl]-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-methanesulfonyl-4-(piperidin-3-yl)-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}pyrimidine
methyl 3-({imidazo[2,1-b][1,3]thiazol-6-ylformamido}methyl)-5-[(2E)-3-phenylprop-2-enamido]benzoate
4-cyclopentyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]pyrimidin-2-amine
2,6-difluoro-4-methoxy-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-3,4-dimethoxy-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
2-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{2-[(pyridin-3-yl)amino]ethyl}cyclopentane-1,3-dicarboxamide
4-[4-(4-fluorophenyl)-4-oxobutyl]-1-(3-methoxyphenyl)piperazin-2-one