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2-(methoxymethyl)-6-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
(1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-yl)methanamine
1-[(3-methoxyphenyl)methyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
7-(cyclopropylmethyl)-2-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{3-[(pyridin-3-yl)amino]propyl}urea
8-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(2S,4R)-4-amino-1-(1,1-dioxo-1λ6-thiane-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
3-(1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
N-(3-methoxypropyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
ethyl 5-{6-amino-5-cyano-4-[5-(hydroxymethyl)furan-2-yl]pyridin-2-yl}-2-methylfuran-3-carboxylate
1-(2-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)piperidin-4-ol
[4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methanol
1-(2-chloro-5-sulfamoylphenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
methyl 1-methyl-2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-1H-1,3-benzodiazole-5-carboxylate
(2R)-2-[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]-2-phenylethan-1-ol
1-[benzyl(methyl)amino]-3-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-{1-[2-(4-fluorobenzenesulfonyl)ethyl]-1H-imidazol-2-yl}quinoline
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-[(pyridin-4-ylmethyl)amino]benzamide
1-(cyclohex-1-ene-1-carbonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
4-(3-methyl-1H-1,2,4-triazol-5-yl)-N-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}piperidine-1-carboxamide
3-{2-[(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
propan-2-yl 3-[(3-carbamoylphenyl)methyl]pyrrolidine-1-carboxylate
N-(1-benzofuran-2-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-[(1R,3S,3aS,6aR)-3-[4-ethoxy-3-(hydroxymethyl)phenyl]-1-(hydroxymethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
4-hydroxy-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(benzylsulfamoyl)[(5-ethylpyridin-2-yl)methyl]methylamine
3-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[1-(4-methylpiperazin-1-yl)propan-2-yl]amino}-1-(4-methylpiperidin-1-yl)propan-1-one
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-methoxy-N-({1-[(3,4,5-trifluorophenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
4-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperidine-1-carboxamide
N-{[7-fluoro-5-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
3,5-dimethyl-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]adamantane-1-carboxamide
(3S,4S)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridine-4-carbonyl)pyrrolidin-3-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methyl-1,3-oxazole-4-carboxamide
(1S,3R)-N1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
3-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}sulfonyl)pyridine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
5-{[2-(2-methoxyphenyl)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(cyclohex-1-ene-1-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
5-ethyl-2-[3-(2-methoxybenzoyl)piperidin-1-yl]pyrimidine
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-oxo-2-phenylacetamide
methyl 2-[3-methyl-2-oxo-4-(quinolin-4-ylmethyl)piperazin-1-yl]acetate
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
9-[(2S)-2-(methylamino)propanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-5,6-dimethylpyridine-3-carboxamide
7-(5-methylthiophen-2-yl)-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol