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N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(2-ethylpyrimidin-4-yl)methyl]methylamine
pyridin-2-yl({1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-yl})methanol
5-{[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,3-oxazolidin-2-one
(2E)-3-(2-chlorophenyl)-1-{4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}prop-2-en-1-one
2-cyclohexyl-6-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1,3-benzoxazole
3-(6-chloro-2-methylpyridin-3-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]urea
2-(4-methylpentyl)-4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]morpholine
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-methylquinoline-4-carboxamide
1-{[3-(4-chlorophenyl)-1,2-oxazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
methyl (2R,4S)-1-{[3-(benzyloxy)phenyl]methyl}-4-hydroxypiperidine-2-carboxylate
(3S,4S)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-(4-chlorophenyl)-5-methyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
N,5-dimethyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-methanesulfonyl-N-propyl-N-(pyridin-3-ylmethyl)benzamide
6-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzothiazol-2-one
9-[(6-ethoxypyridin-3-yl)methyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
[2-(azepan-1-yl)ethyl](methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
1-[(2E)-2-methylbut-2-en-1-yl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
4-[(2S,4R,6S)-4-acetamido-6-(2-phenylethyl)oxan-2-yl]benzoic acid
6-methyl-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)(oxolan-2-ylmethyl)amine
3-(oxolan-3-yl)-5-(1H-pyrazol-3-yl)-1-{[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-1,2,4-triazole
2-(1-benzofuran-2-ylmethyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2,2-dimethylpropyl}morpholine
2-[(4-methoxyphenyl)methyl]-4-(3-methylthiophene-2-carbonyl)morpholine
3-acetyl-N-[(2-chloro-4-fluorophenyl)methyl]-1H-pyrazole-5-carboxamide
1-(furan-3-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-({[1-(2-carbamoylethyl)-1H-indol-3-yl]methyl}amino)-N-ethylpiperidine-1-carboxamide
4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-2-(1,2-oxazol-5-yl)phenol
3-[({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}amino)methyl]piperidin-3-ol
1-methyl-3-(2-methylpropyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
4-hydroxy-N-(2-phenoxyethyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]benzamide
2-{4-[6-amino-5-cyano-4-(4,5-dimethylfuran-2-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
2-{4-[(E)-2-cyclohexylethenyl]-3,5-dimethyl-1H-pyrazol-1-yl}acetamide
2-(2,4-dichlorophenoxy)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
5-(azocane-1-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
N-cyclopropyl-3-(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-3-yl)propanamide
6-methyl-3-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}-4H-chromen-4-one
4-methoxy-N-(oxolan-3-yl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
4-chloro-5-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N'-({1-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl}methyl)ethanediamide
(1S,9R)-11-[5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(2-methylphenyl)methyl]amino}methyl)piperidin-2-one